Assay context summary

Assay context

101 activity records
Activity compounds and values

Activity records

101 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C030428
IC50-=100-200nM---CFPAC-1WO2026061475A1PGDB_A000002PGDB_C030428PGDB_AS000179View
2D structure for PGDB_C030373
IC50-<=1nM---CFPAC-1WO2026061475A1PGDB_A000011PGDB_C030373PGDB_AS000179View
2D structure for PGDB_C030299
IC50-=20-30nM---CFPAC-1WO2026061475A1PGDB_A000052PGDB_C030299PGDB_AS000179View
2D structure for PGDB_C030405
IC50-=200-500nM---CFPAC-1WO2026061475A1PGDB_A000061PGDB_C030405PGDB_AS000179View
2D structure for PGDB_C030392
IC50-=200-500nM---CFPAC-1WO2026061475A1PGDB_A000155PGDB_C030392PGDB_AS000179View
2D structure for PGDB_C030380
IC50-<=1nM---CFPAC-1WO2026061475A1PGDB_A000324PGDB_C030380PGDB_AS000179View
2D structure for PGDB_C030422
IC50-<=1nM---CFPAC-1WO2026061475A1PGDB_A000458PGDB_C030422PGDB_AS000179View
2D structure for PGDB_C030358
IC50-=700-900nM---CFPAC-1WO2026061475A1PGDB_A000596PGDB_C030358PGDB_AS000179View
2D structure for PGDB_C030301
IC50-=200-500nM---CFPAC-1WO2026061475A1PGDB_A000620PGDB_C030301PGDB_AS000179View
2D structure for PGDB_C030434
IC50-=200-500nM---CFPAC-1WO2026061475A1PGDB_A000817PGDB_C030434PGDB_AS000179View
2D structure for PGDB_C030378
IC50-<=1nM---CFPAC-1WO2026061475A1PGDB_A000916PGDB_C030378PGDB_AS000179View
2D structure for PGDB_C030410
IC50-=700-900nM---CFPAC-1WO2026061475A1PGDB_A000918PGDB_C030410PGDB_AS000179View
2D structure for PGDB_C030377
IC50-=10-20nM---CFPAC-1WO2026061475A1PGDB_A001026PGDB_C030377PGDB_AS000179View
2D structure for PGDB_C030389
IC50-=500-700nM---CFPAC-1WO2026061475A1PGDB_A001220PGDB_C030389PGDB_AS000179View
2D structure for PGDB_C030387
IC50-=5-10nM---CFPAC-1WO2026061475A1PGDB_A001332PGDB_C030387PGDB_AS000179View
2D structure for PGDB_C030404
IC50-=10-20nM---CFPAC-1WO2026061475A1PGDB_A001404PGDB_C030404PGDB_AS000179View
2D structure for PGDB_C030408
IC50-=10-20nM---CFPAC-1WO2026061475A1PGDB_A001466PGDB_C030408PGDB_AS000179View
2D structure for PGDB_C030289
IC50-=50-100nM---CFPAC-1WO2026061475A1PGDB_A001634PGDB_C030289PGDB_AS000179View
2D structure for PGDB_C030406
IC50-=200-500nM---CFPAC-1WO2026061475A1PGDB_A001745PGDB_C030406PGDB_AS000179View
2D structure for PGDB_C030437
IC50-=500-700nM---CFPAC-1WO2026061475A1PGDB_A001775PGDB_C030437PGDB_AS000179View