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Nc1nnc(-c2cc(F)ccc2O)cc1N1CC2CCC(C1)N2c1ccc(N2CCN(Cc3ccc(N4CCC(=O)NC4=O)cc3)CC2)cc1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 700-900 | nM | - | — | - | - | CFPAC-1 | WO2026061475A1 | PGDB_A000596 | PGDB_C030358 | PGDB_AS000179 | View | |
| IC50 | - | = | 500-700 | nM | - | — | - | - | A375 | WO2026061475A1 | PGDB_A078225 | PGDB_C030358 | PGDB_AS002441 | View | |
| IC50 | - | = | 200-500 | nM | - | — | - | - | H1944 | WO2026061475A1 | PGDB_A078930 | PGDB_C030358 | PGDB_AS001924 | View | |
| IC50 | - | = | 200-500 | nM | - | — | - | - | H2126 | WO2026061475A1 | PGDB_A081599 | PGDB_C030358 | PGDB_AS001417 | View |