Loading compound
Loading detail record from the SQLite release...
Compound
PGDB_C030399
9 activity records1 related patents
2D structure
Nc1cc2c(cc1SC1CC3CN(CC4CCN(c5ccc(N6C7CCC6CN(c6cc(-c8cc(F)ccc8O)nnc6N)C7)cc5)CC4)CC3C1)CN(C1CCC(=O)NC1=O)C2=OCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 50-100 | nM | - | — | - | - | A549 | WO2026061475A1 | PGDB_A004208 | PGDB_C030399 | PGDB_AS000757 | View |
| IC50 | - | = | 10-20 | nM | - | — | - | - | CFPAC-1 | WO2026061475A1 | PGDB_A004530 | PGDB_C030399 | PGDB_AS000179 | View |
| IC50 | - | = | 10-20 | nM | - | — | - | - | H838 | WO2026061475A1 | PGDB_A004619 | PGDB_C030399 | PGDB_AS000282 | View |
| % Degradation | - | <= | 50 | % | Concentration series: 500 nM, 50 nM | - | SMARCA4 | - | MV-4-11 | WO2026061475A1 | PGDB_A079273 | PGDB_C030399 | PGDB_AS002340 | View |
| IC50 | - | = | 100-200 | nM | - | — | - | - | BT549 | WO2026061475A1 | PGDB_A080796 | PGDB_C030399 | PGDB_AS002259 | View |
| % Degradation | - | <= | 50 | % | Concentration series: 500 nM, 50 nM | - | SMARCA2 | - | MV-4-11 | WO2026061475A1 | PGDB_A081508 | PGDB_C030399 | PGDB_AS002335 | View |