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Compound
PGDB_C030413
9 activity records1 related patents
2D structure
Nc1nnc(-c2cc(F)ccc2O)cc1N1CC2CCC(C1)N2c1ccc(N2CCN(CN3CCN(Nc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)cc1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 900-1000 | nM | - | — | - | - | H1944 | WO2026061475A1 | PGDB_A002356 | PGDB_C030413 | PGDB_AS001924 | View |
| IC50 | - | = | 1-5 | nM | - | — | - | - | H838 | WO2026061475A1 | PGDB_A003480 | PGDB_C030413 | PGDB_AS000282 | View |
| IC50 | - | = | 200-500 | nM | - | — | - | - | CFPAC-1 | WO2026061475A1 | PGDB_A004359 | PGDB_C030413 | PGDB_AS000179 | View |
| IC50 | - | = | 1-5 | nM | - | — | - | - | BT549 | WO2026061475A1 | PGDB_A005350 | PGDB_C030413 | PGDB_AS002259 | View |
| IC50 | - | = | 200-500 | nM | - | — | - | - | A549 | WO2026061475A1 | PGDB_A005826 | PGDB_C030413 | PGDB_AS000757 | View |
| % Degradation | - | <= | 50 | % | Concentration series: 500 nM, 50 nM | - | SMARCA4 | - | MV-4-11 | WO2026061475A1 | PGDB_A078167 | PGDB_C030413 | PGDB_AS002340 | View |
| % Degradation | - | <= | 50 | % | Concentration series: 500 nM, 50 nM | - | SMARCA2 | - | MV-4-11 | WO2026061475A1 | PGDB_A078978 | PGDB_C030413 | PGDB_AS002335 | View |