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O=C1CCN(N2C(=O)c3cccc(N4CCC(CN5CCN(c6ccc7cc(-c8ccccc8O)nnc7c6)CC5)CC4)c3C2=O)C(=O)N1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | <= | 1 | nM | - | — | - | - | CFPAC-1 | WO2026061475A1 | PGDB_A000458 | PGDB_C030422 | PGDB_AS000179 | View | |
| IC50 | - | = | 100-200 | nM | - | — | - | - | BT549 | WO2026061475A1 | PGDB_A000714 | PGDB_C030422 | PGDB_AS002259 | View | |
| IC50 | - | = | 200-500 | nM | - | — | - | - | H2126 | WO2026061475A1 | PGDB_A003237 | PGDB_C030422 | PGDB_AS001417 | View | |
| IC50 | - | <= | 1 | nM | - | — | - | - | H838 | WO2026061475A1 | PGDB_A005135 | PGDB_C030422 | PGDB_AS000282 | View |