Loading compound
Loading detail record from the SQLite release...
Compound
PGDB_C032314
4 activity records1 related patents
2D structure
COC1(C(=O)N(C)C2CCN([C@@H]3COC4(CCN(c5cc(F)c([C@H]6CCC(=O)NC6=O)c(F)c5)CC4)C3)CC2)CCN(c2cnnc(-c3ccccc3O)c2)CC1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | = | 4.42 | nM | - | — | SMARCA2 | - | Calu-6 | WO2026128580A1 | PGDB_A000735 | PGDB_C032314 | PGDB_AS002506 | View |
| Dmax | - | = | 54.51 | % | - | 5 min | SMARCA4 | - | Calu-6 | WO2026128580A1 | PGDB_A005335 | PGDB_C032314 | PGDB_AS002111 | View |
| DC50 | - | = | 174.83 | nM | - | — | SMARCA4 | - | Calu-6 | WO2026128580A1 | PGDB_A080837 | PGDB_C032314 | PGDB_AS001413 | View |
| Dmax | - | = | 87.76 | % | - | - | SMARCA2 | - | Calu-6 | WO2026128580A1 | PGDB_A081347 | PGDB_C032314 | PGDB_AS002073 | View |