Assay

PGDB_AS002506

System: cell_basedTarget: SMARCA2Cell line: Calu-6
Assay context summary

Assay context

179 activity records
Assay family% Degradation
Systemcell_based
ReadoutDC50
TargetSMARCA2
E3Not specified
Cell lineCalu-6
OrganismHomo sapiens
Activity compounds and values

Activity records

179 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C032383
DC50-=4.88nM-—SMARCA2-Calu-6WO2026128580A1PGDB_A000162PGDB_C032383PGDB_AS002506View
2D structure for PGDB_C032416
DC50-=0.9nM-—SMARCA2-Calu-6WO2026128580A1PGDB_A000241PGDB_C032416PGDB_AS002506View
2D structure for PGDB_C032426
DC50-=18.3nM-—SMARCA2-Calu-6WO2026128580A1PGDB_A000330PGDB_C032426PGDB_AS002506View
2D structure for PGDB_C032334
DC50-=4.82nM-—SMARCA2-Calu-6WO2026128580A1PGDB_A000341PGDB_C032334PGDB_AS002506View
2D structure for PGDB_C032364
DC50-=8.78nM-—SMARCA2-Calu-6WO2026128580A1PGDB_A000351PGDB_C032364PGDB_AS002506View
2D structure for PGDB_C032367
DC50-=3.24nM-—SMARCA2-Calu-6WO2026128580A1PGDB_A000446PGDB_C032367PGDB_AS002506View
2D structure for PGDB_C032382
DC50-=7.04nM-—SMARCA2-Calu-6WO2026128580A1PGDB_A000554PGDB_C032382PGDB_AS002506View
2D structure for PGDB_C032333
DC50-=4.65nM-—SMARCA2-Calu-6WO2026128580A1PGDB_A000636PGDB_C032333PGDB_AS002506View
2D structure for PGDB_C032399
DC50-=7.39nM-—SMARCA2-Calu-6WO2026128580A1PGDB_A000730PGDB_C032399PGDB_AS002506View
2D structure for PGDB_C032314
DC50-=4.42nM-—SMARCA2-Calu-6WO2026128580A1PGDB_A000735PGDB_C032314PGDB_AS002506View
2D structure for PGDB_C032266
DC50-=15.6nM-—SMARCA2-Calu-6WO2026128580A1PGDB_A000737PGDB_C032266PGDB_AS002506View
2D structure for PGDB_C032396
DC50-=3.6nM-—SMARCA2-Calu-6WO2026128580A1PGDB_A000819PGDB_C032396PGDB_AS002506View
2D structure for PGDB_C032323
DC50-=1.57nM-—SMARCA2-Calu-6WO2026128580A1PGDB_A000936PGDB_C032323PGDB_AS002506View
2D structure for PGDB_C032424
DC50-=5.85nM-—SMARCA2-Calu-6WO2026128580A1PGDB_A000963PGDB_C032424PGDB_AS002506View
2D structure for PGDB_C032310
DC50-=8.14nM-—SMARCA2-Calu-6WO2026128580A1PGDB_A000999PGDB_C032310PGDB_AS002506View
2D structure for PGDB_C032357
DC50-=2.08nM-—SMARCA2-Calu-6WO2026128580A1PGDB_A001039PGDB_C032357PGDB_AS002506View
2D structure for PGDB_C032279
DC50-=12.08nM-—SMARCA2-Calu-6WO2026128580A1PGDB_A001043PGDB_C032279PGDB_AS002506View
2D structure for PGDB_C032293
DC50-=2.27nM-—SMARCA2-Calu-6WO2026128580A1PGDB_A001061PGDB_C032293PGDB_AS002506View
2D structure for PGDB_C032277
DC50-=21.78nM-—SMARCA2-Calu-6WO2026128580A1PGDB_A001086PGDB_C032277PGDB_AS002506View
2D structure for PGDB_C032400
DC50-=6.75nM-—SMARCA2-Calu-6WO2026128580A1PGDB_A001089PGDB_C032400PGDB_AS002506View
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