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CCN(C(=O)C1(OC)CCN(c2cnnc(-c3ccccc3O)c2)CC1)C1CCN(CCC2(F)CCN(c3ccc([C@H]4CCC(=O)NC4=O)c(F)c3)CC2)CC1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 56.27 | % | - | 5 min | SMARCA4 | - | Calu-6 | WO2026128580A1 | PGDB_A000204 | PGDB_C032376 | PGDB_AS002111 | View | |
| DC50 | - | = | 99.7 | nM | - | — | SMARCA4 | - | Calu-6 | WO2026128580A1 | PGDB_A000782 | PGDB_C032376 | PGDB_AS001413 | View | |
| DC50 | - | = | 2.65 | nM | - | — | SMARCA2 | - | Calu-6 | WO2026128580A1 | PGDB_A001633 | PGDB_C032376 | PGDB_AS002506 | View | |
| Dmax | - | = | 96.1 | % | - | - | SMARCA2 | - | Calu-6 | WO2026128580A1 | PGDB_A003548 | PGDB_C032376 | PGDB_AS002073 | View |