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Compound
PGDB_C032383
8 activity records1 related patents
2D structure
COCC1(C(=O)N(C2CC2)C2CCN(CCC3CCN(c4ccc([C@@H]5CCC(=O)NC5=O)cc4)CC3)CC2)CCN(c2cnnc(-c3ccccc3O)c2)CC1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | = | 4.88 | nM | - | — | SMARCA2 | - | Calu-6 | WO2026128580A1 | PGDB_A000162 | PGDB_C032383 | PGDB_AS002506 | View |
| DC50 | - | = | 1.81 | nM | - | — | SMARCA2 | - | Calu-6 | WO2026128580A1 | PGDB_A002719 | PGDB_C032383 | PGDB_AS002506 | View |
| Dmax | - | = | 87.76 | % | - | - | SMARCA2 | - | Calu-6 | WO2026128580A1 | PGDB_A005543 | PGDB_C032383 | PGDB_AS002073 | View |
| Dmax | - | = | 92.49 | % | - | - | SMARCA2 | - | Calu-6 | WO2026128580A1 | PGDB_A005774 | PGDB_C032383 | PGDB_AS002073 | View |
| DC50 | - | = | 1000 | nM | - | — | SMARCA4 | - | Calu-6 | WO2026128580A1 | PGDB_A078156 | PGDB_C032383 | PGDB_AS001413 | View |
| DC50 | - | = | 1000 | nM | - | — | SMARCA4 | - | Calu-6 | WO2026128580A1 | PGDB_A078876 | PGDB_C032383 | PGDB_AS001413 | View |
| Dmax | - | = | 21.95 | % | - | 5 min | SMARCA4 | - | Calu-6 | WO2026128580A1 | PGDB_A079567 | PGDB_C032383 | PGDB_AS002111 | View |
| Dmax | - | = | 33.94 | % | - | 5 min | SMARCA4 | - | Calu-6 | WO2026128580A1 | PGDB_A081809 | PGDB_C032383 | PGDB_AS002111 | View |