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Compound
PGDB_C032399
4 activity records1 related patents
2D structure
CCC1(C(=O)N(C)C2CCN(CCC3CCN(c4ccc([C@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)CCN(c2cnnc(-c3ccccc3O)c2)CC1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 88.35 | % | - | - | SMARCA2 | - | Calu-6 | WO2026128580A1 | PGDB_A000057 | PGDB_C032399 | PGDB_AS002073 | View |
| DC50 | - | = | 7.39 | nM | - | — | SMARCA2 | - | Calu-6 | WO2026128580A1 | PGDB_A000730 | PGDB_C032399 | PGDB_AS002506 | View |
| DC50 | - | = | 135 | nM | - | — | SMARCA4 | - | Calu-6 | WO2026128580A1 | PGDB_A002252 | PGDB_C032399 | PGDB_AS001413 | View |
| Dmax | - | = | 60.64 | % | - | 5 min | SMARCA4 | - | Calu-6 | WO2026128580A1 | PGDB_A080175 | PGDB_C032399 | PGDB_AS002111 | View |