Loading compound
Loading detail record from the SQLite release...
Loading detail record from the SQLite release...
COCCN(C(=O)[C@H]1[C@@H]2CC[C@H]1CN(c1cnnc(-c3ccccc3O)c1)C2)C1CCN(CCC2CCN(c3ccc([C@@H]4CCC(=O)NC4=O)c(F)c3)CC2)CC1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 84.53 | % | - | - | SMARCA2 | - | Calu-6 | WO2026128580A1 | PGDB_A000053 | PGDB_C032432 | PGDB_AS002073 | View | |
| DC50 | - | = | 1000 | nM | - | — | SMARCA4 | - | Calu-6 | WO2026128580A1 | PGDB_A000937 | PGDB_C032432 | PGDB_AS001413 | View | |
| DC50 | - | = | 23 | nM | - | — | SMARCA2 | - | Calu-6 | WO2026128580A1 | PGDB_A003172 | PGDB_C032432 | PGDB_AS002506 | View | |
| Dmax | - | = | 15.1 | % | - | 5 min | SMARCA4 | - | Calu-6 | WO2026128580A1 | PGDB_A078102 | PGDB_C032432 | PGDB_AS002111 | View |