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Compound
PGDB_C032441
8 activity records1 related patents
2D structure
CCN(C(=O)C1(OC)CCN(c2cnnc(-c3ccccc3O)c2)CC1)C1CCN(CCC2(F)CCN(c3ccc([C@H]4CCC(=O)NC4=O)cc3)CC2)CC1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | = | 10000 | nM | - | — | SMARCA4 | - | Calu-6 | WO2026128580A1 | PGDB_A000238 | PGDB_C032441 | PGDB_AS001413 | View |
| Dmax | - | = | 84.34 | % | - | - | SMARCA2 | - | Calu-6 | WO2026128580A1 | PGDB_A000603 | PGDB_C032441 | PGDB_AS002073 | View |
| DC50 | - | = | 5.11 | nM | - | — | SMARCA2 | - | Calu-6 | WO2026128580A1 | PGDB_A002114 | PGDB_C032441 | PGDB_AS002506 | View |
| Dmax | - | = | 38.38 | % | - | 5 min | SMARCA4 | - | Calu-6 | WO2026128580A1 | PGDB_A002312 | PGDB_C032441 | PGDB_AS002111 | View |
| Dmax | - | = | 29.48 | % | - | 5 min | SMARCA4 | - | Calu-6 | WO2026128580A1 | PGDB_A003535 | PGDB_C032441 | PGDB_AS002111 | View |
| DC50 | - | = | 1000 | nM | - | — | SMARCA4 | - | Calu-6 | WO2026128580A1 | PGDB_A005868 | PGDB_C032441 | PGDB_AS001413 | View |
| DC50 | - | = | 6.64 | nM | - | — | SMARCA2 | - | Calu-6 | WO2026128580A1 | PGDB_A079793 | PGDB_C032441 | PGDB_AS002506 | View |
| Dmax | - | = | 90.38 | % | - | - | SMARCA2 | - | Calu-6 | WO2026128580A1 | PGDB_A081186 | PGDB_C032441 | PGDB_AS002073 | View |