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Compound
PGDB_C032442
8 activity records1 related patents
2D structure
COC1(C(=O)N2CCC3(CC2)CCN([C@H]2COC4(CCN(c5ccc([C@H]6CCC(=O)NC6=O)cc5)CC4)C2)C3)CCN(c2cnnc(-c3ccccc3O)c2)CC1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | = | 41.3 | nM | - | — | SMARCA4 | - | Calu-6 | WO2026128580A1 | PGDB_A000682 | PGDB_C032442 | PGDB_AS001413 | View |
| DC50 | - | = | 7.35 | nM | - | — | SMARCA2 | - | Calu-6 | WO2026128580A1 | PGDB_A004277 | PGDB_C032442 | PGDB_AS002506 | View |
| Dmax | - | = | 61.8 | % | - | 5 min | SMARCA4 | - | Calu-6 | WO2026128580A1 | PGDB_A005321 | PGDB_C032442 | PGDB_AS002111 | View |
| DC50 | - | = | 7.35 | nM | - | — | SMARCA2 | - | Calu-6 | WO2026128580A1 | PGDB_A006328 | PGDB_C032442 | PGDB_AS002506 | View |
| Dmax | - | = | 61.8 | % | - | 5 min | SMARCA4 | - | Calu-6 | WO2026128580A1 | PGDB_A078382 | PGDB_C032442 | PGDB_AS002111 | View |
| Dmax | - | = | 82.68 | % | - | - | SMARCA2 | - | Calu-6 | WO2026128580A1 | PGDB_A079163 | PGDB_C032442 | PGDB_AS002073 | View |
| Dmax | - | = | 82.68 | % | - | - | SMARCA2 | - | Calu-6 | WO2026128580A1 | PGDB_A079704 | PGDB_C032442 | PGDB_AS002073 | View |
| DC50 | - | = | 41.3 | nM | - | — | SMARCA4 | - | Calu-6 | WO2026128580A1 | PGDB_A079999 | PGDB_C032442 | PGDB_AS001413 | View |