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Patent
CA3173658A1
2 compounds10 activity records5 assays
Patent summary
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | ||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
 | IC50 | - | = | 97-204 | nM | - | — | IKZF1 | - | NCI-H929 | PGDB_A009780 | PGDB_C009601 | PGDB_AS001574 | View |
 | IC50 | - | = | 0.033-0.149 | nM | - | — | IKZF1 | - | NCI-H929 | PGDB_A020043 | PGDB_C006053 | PGDB_AS001574 | View |
| IC50 | - | = | 0.27 | nM | - | — | IKZF1 | - | - | PGDB_A024467 | PGDB_C006053 | PGDB_AS000746 | View |
| IC50 | - | = | 0.071 | nM | - | — | IKZF1 | - | NCI-H929 | PGDB_A033512 | PGDB_C006053 | PGDB_AS000269 | View |
| Emax | - | = | 22.4 | % | 1 uM | 55.7 ± 6.0 | 22.4 ± 3.1 | IKZF1 | - | - | PGDB_A052717 | PGDB_C006053 | PGDB_AS001198 | View |
| Emax | - | = | 15.6 | % | 1 uM | 97 - 204 | 0.033 - 0.149 | IKZF1 | - | NCI-H929 | PGDB_A056536 | PGDB_C009601 | PGDB_AS002447 | View |
| Emax | - | = | 55.7 | % | 1 uM | 55.7 ± 6.0 | 22.4 ± 3.1 | IKZF1 | - | - | PGDB_A058737 | PGDB_C009601 | PGDB_AS001198 | View |
| IC50 | - | = | 141 | nM | - | — | IKZF1 | - | NCI-H929 | PGDB_A059289 | PGDB_C009601 | PGDB_AS000269 | View |
| Emax | - | = | 4 | % | 1 uM | 97 - 204 | 0.033 - 0.149 | IKZF1 | - | NCI-H929 | PGDB_A063927 | PGDB_C006053 | PGDB_AS002447 | View |
| IC50 | - | > | 833 | nM | - | — | IKZF1 | - | - | PGDB_A076893 | PGDB_C009601 | PGDB_AS000746 | View |