Assay
PGDB_AS000080
System: cell_basedCell line: MV-4-11
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | BTK | - | MV-4-11 | CN116239566A | PGDB_A016007 | PGDB_C025815 | PGDB_AS000080 | View | |
| IC50 | - | = | 100-500 | nM | - | — | BTK | - | MV-4-11 | CN116239566A | PGDB_A034707 | PGDB_C025811 | PGDB_AS000080 | View | |
| IC50 | - | = | 50-100 | nM | - | — | BTK | - | MV-4-11 | CN116239566A | PGDB_A038647 | PGDB_C025803 | PGDB_AS000080 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | MV-4-11 | CN116239566A | PGDB_A064070 | PGDB_C015982 | PGDB_AS000080 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | MV-4-11 | CN116239566A | PGDB_A066724 | PGDB_C025807 | PGDB_AS000080 | View |