Assay

PGDB_AS000168

System: cell_basedTarget: GSPT1Cell line: HEK293
Assay context summary

Assay context

7 activity records
Assay family% Degradation
Systemcell_based
ReadoutEC50
TargetGSPT1
E3CRBN
Cell lineHEK293
OrganismHomo sapiens
Technologyluminescence
Activity compounds and values

Activity records

7 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C001430
EC50-<1uM-—GSPT1CRBNHEK293WO2022066835A1PGDB_A020667PGDB_C001430PGDB_AS000168View
2D structure for PGDB_C001361
EC50-<1uM-—GSPT1CRBNHEK293WO2022066835A1PGDB_A045625PGDB_C001361PGDB_AS000168View
2D structure for PGDB_C019545
EC50-<1uM-—GSPT1CRBNHEK293WO2022066835A1PGDB_A046409PGDB_C019545PGDB_AS000168View
2D structure for PGDB_C019590
EC50-<1uM-—GSPT1CRBNHEK293WO2022066835A1PGDB_A047729PGDB_C019590PGDB_AS000168View
2D structure for PGDB_C021183
EC50-<1uM-—GSPT1CRBNHEK293WO2022066835A1PGDB_A051008PGDB_C021183PGDB_AS000168View
2D structure for PGDB_C019591
EC50-<1uM-—GSPT1CRBNHEK293WO2022066835A1PGDB_A056592PGDB_C019591PGDB_AS000168View
2D structure for PGDB_C019590
EC50-<1uM-—GSPT1CRBNHEK293WO2022066835A1PGDB_A072775PGDB_C019590PGDB_AS000168View
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