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SIMM · NJU
Assay
PGDB_AS000265
System: cell_based
Cell line: A2058
Assay context summary
Assay context
38 activity records
Assay family
viability
System
cell_based
Readout
IC50
E3
Not specified
Cell line
A2058
Technology
luminescence
Detection target
cell_proliferation
Activity compounds and values
Activity records
38 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
IC50
-
=
0.4
nM
-
—
PDE3A
-
A2058
CN120265631A
PGDB_A007087
PGDB_C007100
PGDB_AS000265
View
IC50
-
=
31.9
nM
-
—
PDE3A
-
A2058
CN120265631A
PGDB_A008152
PGDB_C007098
PGDB_AS000265
View
IC50
-
=
5.2
nM
-
—
PDE3A
-
A2058
CN120265631A
PGDB_A009242
PGDB_C007118
PGDB_AS000265
View
IC50
-
=
2.7
nM
-
—
PDE3A
-
A2058
CN120265631A
PGDB_A009411
PGDB_C007108
PGDB_AS000265
View
IC50
-
=
1.1
nM
-
—
PDE3A
-
A2058
CN120265631A
PGDB_A009917
PGDB_C007085
PGDB_AS000265
View
IC50
-
=
5.2
nM
-
—
PDE3A
-
A2058
CN120265631A
PGDB_A012133
PGDB_C007119
PGDB_AS000265
View
IC50
-
=
1.2
nM
-
—
PDE3A
-
A2058
CN120265631A
PGDB_A014766
PGDB_C007066
PGDB_AS000265
View
IC50
-
=
0.19
nM
-
—
PDE3A
-
A2058
CN120265631A
PGDB_A020190
PGDB_C007117
PGDB_AS000265
View
IC50
-
=
2
nM
-
—
PDE3A
-
A2058
CN120265631A
PGDB_A024839
PGDB_C007149
PGDB_AS000265
View
IC50
-
=
1
nM
-
—
PDE3A
-
A2058
CN120265631A
PGDB_A026413
PGDB_C007134
PGDB_AS000265
View
IC50
-
=
1.7
nM
-
—
PDE3A
-
A2058
CN120265631A
PGDB_A026737
PGDB_C007096
PGDB_AS000265
View
IC50
-
=
8
nM
-
—
PDE3A
-
A2058
CN120265631A
PGDB_A031168
PGDB_C007137
PGDB_AS000265
View
IC50
-
=
7.5
nM
-
—
PDE3A
-
A2058
CN120265631A
PGDB_A034905
PGDB_C007072
PGDB_AS000265
View
IC50
-
=
0.3
nM
-
—
PDE3A
-
A2058
CN120265631A
PGDB_A041452
PGDB_C007116
PGDB_AS000265
View
IC50
-
=
0.4
nM
-
—
PDE3A
-
A2058
CN120265631A
PGDB_A044043
PGDB_C007139
PGDB_AS000265
View
IC50
-
=
3.3
nM
-
—
PDE3A
-
A2058
CN120265631A
PGDB_A045535
PGDB_C007136
PGDB_AS000265
View
IC50
-
=
0.29
nM
-
—
PDE3A
-
A2058
CN120265631A
PGDB_A046311
PGDB_C007101
PGDB_AS000265
View
IC50
-
=
0.17
nM
-
—
PDE3A
-
A2058
CN120265631A
PGDB_A046333
PGDB_C007140
PGDB_AS000265
View
IC50
-
=
1.2
nM
-
—
PDE3A
-
A2058
CN120265631A
PGDB_A048366
PGDB_C007094
PGDB_AS000265
View
IC50
-
=
11.9
nM
-
—
PDE3A
-
A2058
CN120265631A
PGDB_A048598
PGDB_C007093
PGDB_AS000265
View