Assay context summary

Assay context

38 activity records
Activity compounds and values

Activity records

38 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C007100
IC50-=0.4nM-PDE3A-A2058CN120265631APGDB_A007087PGDB_C007100PGDB_AS000265View
2D structure for PGDB_C007098
IC50-=31.9nM-PDE3A-A2058CN120265631APGDB_A008152PGDB_C007098PGDB_AS000265View
2D structure for PGDB_C007118
IC50-=5.2nM-PDE3A-A2058CN120265631APGDB_A009242PGDB_C007118PGDB_AS000265View
2D structure for PGDB_C007108
IC50-=2.7nM-PDE3A-A2058CN120265631APGDB_A009411PGDB_C007108PGDB_AS000265View
2D structure for PGDB_C007085
IC50-=1.1nM-PDE3A-A2058CN120265631APGDB_A009917PGDB_C007085PGDB_AS000265View
2D structure for PGDB_C007119
IC50-=5.2nM-PDE3A-A2058CN120265631APGDB_A012133PGDB_C007119PGDB_AS000265View
2D structure for PGDB_C007066
IC50-=1.2nM-PDE3A-A2058CN120265631APGDB_A014766PGDB_C007066PGDB_AS000265View
2D structure for PGDB_C007117
IC50-=0.19nM-PDE3A-A2058CN120265631APGDB_A020190PGDB_C007117PGDB_AS000265View
2D structure for PGDB_C007149
IC50-=2nM-PDE3A-A2058CN120265631APGDB_A024839PGDB_C007149PGDB_AS000265View
2D structure for PGDB_C007134
IC50-=1nM-PDE3A-A2058CN120265631APGDB_A026413PGDB_C007134PGDB_AS000265View
2D structure for PGDB_C007096
IC50-=1.7nM-PDE3A-A2058CN120265631APGDB_A026737PGDB_C007096PGDB_AS000265View
2D structure for PGDB_C007137
IC50-=8nM-PDE3A-A2058CN120265631APGDB_A031168PGDB_C007137PGDB_AS000265View
2D structure for PGDB_C007072
IC50-=7.5nM-PDE3A-A2058CN120265631APGDB_A034905PGDB_C007072PGDB_AS000265View
2D structure for PGDB_C007116
IC50-=0.3nM-PDE3A-A2058CN120265631APGDB_A041452PGDB_C007116PGDB_AS000265View
2D structure for PGDB_C007139
IC50-=0.4nM-PDE3A-A2058CN120265631APGDB_A044043PGDB_C007139PGDB_AS000265View
2D structure for PGDB_C007136
IC50-=3.3nM-PDE3A-A2058CN120265631APGDB_A045535PGDB_C007136PGDB_AS000265View
2D structure for PGDB_C007101
IC50-=0.29nM-PDE3A-A2058CN120265631APGDB_A046311PGDB_C007101PGDB_AS000265View
2D structure for PGDB_C007140
IC50-=0.17nM-PDE3A-A2058CN120265631APGDB_A046333PGDB_C007140PGDB_AS000265View
2D structure for PGDB_C007094
IC50-=1.2nM-PDE3A-A2058CN120265631APGDB_A048366PGDB_C007094PGDB_AS000265View
2D structure for PGDB_C007093
IC50-=11.9nM-PDE3A-A2058CN120265631APGDB_A048598PGDB_C007093PGDB_AS000265View