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O=c1[nH]c2cc3cc(-c4cnn(C(F)F)c4Br)ccc3nc2[nH]1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 1.6 | nM | - | — | PDE3A | - | - | CN120265631A | PGDB_A024753 | PGDB_C007116 | PGDB_AS000140 | View | |
| IC50 | - | = | 0.05 | nM | - | — | PDE3A | - | SK-MEL-3 | CN120265631A | PGDB_A038890 | PGDB_C007116 | PGDB_AS001659 | View | |
| IC50 | - | = | 0.3 | nM | - | — | PDE3A | - | A2058 | CN120265631A | PGDB_A041452 | PGDB_C007116 | PGDB_AS000265 | View |