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O=c1[nH]c2cc3c(nc2[nH]1)CC[C@@H](c1cnn(C(F)F)c1Cl)C3| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 0.4 | nM | - | — | PDE3A | - | A2058 | CN120265631A | PGDB_A007087 | PGDB_C007100 | PGDB_AS000265 | View | |
| IC50 | - | = | 21.77 | nM | - | — | PDE3A | - | - | CN120265631A | PGDB_A017410 | PGDB_C007100 | PGDB_AS000140 | View | |
| IC50 | - | = | 0.5 | nM | - | — | PDE3A | - | SK-MEL-3 | CN120265631A | PGDB_A038346 | PGDB_C007100 | PGDB_AS001659 | View | |
| IC50 | - | = | 0.08 | nM | - | — | PDE3A | - | SK-MEL-3 | CN120265631A | PGDB_A042465 | PGDB_C007100 | PGDB_AS001659 | View | |
| IC50 | - | = | 1.79 | nM | - | — | PDE3A | - | A2058 | CN120265631A | PGDB_A074174 | PGDB_C007100 | PGDB_AS000265 | View |