Assay
PGDB_AS000343
System: cell_basedCell line: NCI-H929
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | <= | 25 | % | 20 uM | 24 h | CSNK1A1 | - | NCI-H929 | AU2020392427A1 | PGDB_A009266 | PGDB_C019025 | PGDB_AS000343 | View | |
| % Degradation | - | <= | 25 | % | 20 uM | 24 h | CSNK1A1 | - | NCI-H929 | AU2020392427A1 | PGDB_A021571 | PGDB_C019016 | PGDB_AS000343 | View | |
| % Degradation | - | <= | 25 | % | 20 uM | 24 h | CSNK1A1 | - | NCI-H929 | AU2020392427A1 | PGDB_A025355 | PGDB_C019028 | PGDB_AS000343 | View | |
| % Degradation | - | <= | 25 | % | 20 uM | 24 h | CSNK1A1 | - | NCI-H929 | AU2020392427A1 | PGDB_A028877 | PGDB_C019040 | PGDB_AS000343 | View | |
| % Degradation | - | <= | 25 | % | 20 uM | 24 h | CSNK1A1 | - | NCI-H929 | AU2020392427A1 | PGDB_A029315 | PGDB_C019027 | PGDB_AS000343 | View | |
| % Degradation | - | <= | 25 | % | 20 uM | 24 h | CSNK1A1 | - | NCI-H929 | AU2020392427A1 | PGDB_A032454 | PGDB_C019029 | PGDB_AS000343 | View | |
| % Degradation | - | <= | 25 | % | 20 uM | 24 h | CSNK1A1 | - | NCI-H929 | AU2020392427A1 | PGDB_A050801 | PGDB_C019014 | PGDB_AS000343 | View | |
| % Degradation | - | <= | 25 | % | 20 uM | 24 h | CSNK1A1 | - | NCI-H929 | AU2020392427A1 | PGDB_A055679 | PGDB_C019020 | PGDB_AS000343 | View | |
| % Degradation | - | <= | 25 | % | 20 uM | 24 h | CSNK1A1 | - | NCI-H929 | AU2020392427A1 | PGDB_A074783 | PGDB_C019017 | PGDB_AS000343 | View |