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CS(=O)(=O)c1cccc(CNc2nc(Nc3ccc(N4CCN(Cc5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6)CC4)cc3)ncc2C(F)(F)F)c1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | SW620 | CN116239566A | PGDB_A029922 | PGDB_C025950 | PGDB_AS001904 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | VCaP | CN116239566A | PGDB_A048395 | PGDB_C025950 | PGDB_AS000495 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | SR | CN116239566A | PGDB_A048594 | PGDB_C025950 | PGDB_AS001780 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | HGC-27 | CN116239566A | PGDB_A062205 | PGDB_C025950 | PGDB_AS001781 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | PC-9 | CN116239566A | PGDB_A063447 | PGDB_C025950 | PGDB_AS001387 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | Mino | CN116239566A | PGDB_A067036 | PGDB_C025950 | PGDB_AS000370 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | CCRF-CEM | CN116239566A | PGDB_A073373 | PGDB_C025950 | PGDB_AS000686 | View |