Assay
PGDB_AS000407
System: biochemicalTarget: CRBN
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 239 | nM | - | — | CRBN | CRBN | - | WO2024125437A1 | PGDB_A030392 | PGDB_C005368 | PGDB_AS000407 | View | |
| IC50 | - | = | 83 | nM | - | — | CRBN | CRBN | - | WO2024125437A1 | PGDB_A039175 | PGDB_C005360 | PGDB_AS000407 | View | |
| IC50 | - | = | 59 | nM | - | — | CRBN | CRBN | - | WO2024125437A1 | PGDB_A040950 | PGDB_C005364 | PGDB_AS000407 | View | |
| IC50 | - | = | 130 | nM | - | — | CRBN | CRBN | - | WO2024125437A1 | PGDB_A042510 | PGDB_C005366 | PGDB_AS000407 | View | |
| IC50 | - | = | 167 | nM | - | — | CRBN | CRBN | - | WO2024125437A1 | PGDB_A042605 | PGDB_C005370 | PGDB_AS000407 | View | |
| IC50 | - | = | 203 | nM | - | — | CRBN | CRBN | - | WO2024125437A1 | PGDB_A051776 | PGDB_C005361 | PGDB_AS000407 | View |