Assay
PGDB_AS000420
System: cell_basedCell line: JeKo-1
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | BTK | - | JeKo-1 | CN116239566A | PGDB_A031896 | PGDB_C025809 | PGDB_AS000420 | View | |
| IC50 | - | = | 50-100 | nM | - | — | BTK | - | JeKo-1 | CN116239566A | PGDB_A045913 | PGDB_C025815 | PGDB_AS000420 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | JeKo-1 | CN116239566A | PGDB_A055550 | PGDB_C025808 | PGDB_AS000420 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | JeKo-1 | CN116239566A | PGDB_A056667 | PGDB_C015982 | PGDB_AS000420 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | JeKo-1 | CN116239566A | PGDB_A064898 | PGDB_C019593 | PGDB_AS000420 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | JeKo-1 | CN116239566A | PGDB_A075596 | PGDB_C025807 | PGDB_AS000420 | View |