Assay
PGDB_AS000469
System: cell_basedCell line: CCRF-CEM
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | BTK | - | CCRF-CEM | CN116239566A | PGDB_A032065 | PGDB_C025813 | PGDB_AS000469 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | CCRF-CEM | CN116239566A | PGDB_A045496 | PGDB_C025807 | PGDB_AS000469 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | CCRF-CEM | CN116239566A | PGDB_A049670 | PGDB_C025806 | PGDB_AS000469 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | CCRF-CEM | CN116239566A | PGDB_A050536 | PGDB_C025808 | PGDB_AS000469 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | CCRF-CEM | CN116239566A | PGDB_A056065 | PGDB_C025814 | PGDB_AS000469 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | CCRF-CEM | CN116239566A | PGDB_A067124 | PGDB_C025803 | PGDB_AS000469 | View |