Assay
PGDB_AS000486
System: cell_basedCell line: THP-1
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
 | IC50 | - | = | 1000-5000 | nM | - | — | BTK | - | THP-1 | CN116239566A | PGDB_A011017 | PGDB_C025813 | PGDB_AS000486 | View |
 | IC50 | - | < | 50 | nM | - | — | BTK | - | THP-1 | CN116239566A | PGDB_A026842 | PGDB_C025806 | PGDB_AS000486 | View |
 | IC50 | - | < | 50 | nM | - | — | BTK | - | THP-1 | CN116239566A | PGDB_A030154 | PGDB_C015982 | PGDB_AS000486 | View |
 | IC50 | - | = | 100-500 | nM | - | — | BTK | - | THP-1 | CN116239566A | PGDB_A035381 | PGDB_C025815 | PGDB_AS000486 | View |
 | IC50 | - | < | 50 | nM | - | — | BTK | - | THP-1 | CN116239566A | PGDB_A036860 | PGDB_C025808 | PGDB_AS000486 | View |
 | IC50 | - | < | 50 | nM | - | — | BTK | - | THP-1 | CN116239566A | PGDB_A039218 | PGDB_C025807 | PGDB_AS000486 | View |
 | IC50 | - | < | 50 | nM | - | — | BTK | - | THP-1 | CN116239566A | PGDB_A059275 | PGDB_C025805 | PGDB_AS000486 | View |