Assay

PGDB_AS000488

System: biochemicalTarget: CRBN
Assay context summary

Assay context

204 activity records
Assay familybiochemical
Systembiochemical
ReadoutEC50
TargetCRBN
E3CRBN
TechnologyHTRF
Activity compounds and values

Activity records

204 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C020245
EC50-=100-1000nM-—CRBNCRBN-WO2025024521A1PGDB_A007359PGDB_C020245PGDB_AS000488View
2D structure for PGDB_C020342
EC50-=100-1000nM-—CRBNCRBN-WO2025024521A1PGDB_A007388PGDB_C020342PGDB_AS000488View
2D structure for PGDB_C026233
EC50-<100nM-—CRBNCRBN-WO2025024521A1PGDB_A007795PGDB_C026233PGDB_AS000488View
2D structure for PGDB_C020445
EC50-=100-1000nM-—CRBNCRBN-WO2025024521A1PGDB_A007937PGDB_C020445PGDB_AS000488View
2D structure for PGDB_C020360
EC50-<100nM-—CRBNCRBN-WO2025024521A1PGDB_A008467PGDB_C020360PGDB_AS000488View
2D structure for PGDB_C020200
EC50-<100nM-—CRBNCRBN-WO2025024521A1PGDB_A008748PGDB_C020200PGDB_AS000488View
2D structure for PGDB_C020412
EC50-=100-1000nM-—CRBNCRBN-WO2025024521A1PGDB_A008769PGDB_C020412PGDB_AS000488View
2D structure for PGDB_C020435
EC50-<100nM-—CRBNCRBN-WO2025024521A1PGDB_A008832PGDB_C020435PGDB_AS000488View
2D structure for PGDB_C020430
EC50-<100nM-—CRBNCRBN-WO2025024521A1PGDB_A009470PGDB_C020430PGDB_AS000488View
2D structure for PGDB_C020358
EC50-<100nM-—CRBNCRBN-WO2025024521A1PGDB_A009564PGDB_C020358PGDB_AS000488View
2D structure for PGDB_C020177
EC50-=100-1000nM-—CRBNCRBN-WO2025024521A1PGDB_A009610PGDB_C020177PGDB_AS000488View
2D structure for PGDB_C020456
EC50-=100-1000nM-—CRBNCRBN-WO2025024521A1PGDB_A009636PGDB_C020456PGDB_AS000488View
2D structure for PGDB_C020455
EC50-=100-1000nM-—CRBNCRBN-WO2025024521A1PGDB_A009747PGDB_C020455PGDB_AS000488View
2D structure for PGDB_C020332
EC50-=100-1000nM-—CRBNCRBN-WO2025024521A1PGDB_A010834PGDB_C020332PGDB_AS000488View
2D structure for PGDB_C020424
EC50-<100nM-—CRBNCRBN-WO2025024521A1PGDB_A011452PGDB_C020424PGDB_AS000488View
2D structure for PGDB_C020196
EC50-=100-1000nM-—CRBNCRBN-WO2025024521A1PGDB_A011733PGDB_C020196PGDB_AS000488View
2D structure for PGDB_C026277
EC50-<100nM-—CRBNCRBN-WO2025024521A1PGDB_A012231PGDB_C026277PGDB_AS000488View
2D structure for PGDB_C020259
EC50-=100-1000nM-—CRBNCRBN-WO2025024521A1PGDB_A012504PGDB_C020259PGDB_AS000488View
2D structure for PGDB_C016406
EC50-=100-1000nM-—CRBNCRBN-WO2025024521A1PGDB_A012961PGDB_C016406PGDB_AS000488View
2D structure for PGDB_C020320
EC50-=100-1000nM-—CRBNCRBN-WO2025024521A1PGDB_A013117PGDB_C020320PGDB_AS000488View
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