PatGlueDB
Search
Browse
Statistics
Contact
Help
·
SIMM · NJU
Assay
PGDB_AS000508
System: cell_based
Target: WIZ
Cell line: HT-1080
Assay context summary
Assay context
115 activity records
Assay family
% Degradation
System
cell_based
Readout
DC50
Target
WIZ
E3
Not specified
Cell line
HT-1080
Organism
Homo sapiens
Technology
luminescence
Activity compounds and values
Activity records
115 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
DC50
-
=
16.6
nM
-
—
WIZ
-
HT-1080
WO2025256460A1
PGDB_A007034
PGDB_C012089
PGDB_AS000508
View
DC50
-
=
44.1
nM
-
—
WIZ
-
HT-1080
WO2025256460A1
PGDB_A007446
PGDB_C012145
PGDB_AS000508
View
DC50
-
=
10.3
nM
-
—
WIZ
-
HT-1080
WO2025256460A1
PGDB_A008228
PGDB_C012090
PGDB_AS000508
View
DC50
-
=
11.9
nM
-
—
WIZ
-
HT-1080
WO2025256460A1
PGDB_A008330
PGDB_C012106
PGDB_AS000508
View
DC50
-
=
23.8
nM
-
—
WIZ
-
HT-1080
WO2025256460A1
PGDB_A010414
PGDB_C012120
PGDB_AS000508
View
DC50
-
=
7.2
nM
-
—
WIZ
-
HT-1080
WO2025256460A1
PGDB_A010941
PGDB_C012150
PGDB_AS000508
View
DC50
-
=
40.2
nM
-
—
WIZ
-
HT-1080
WO2025256460A1
PGDB_A011136
PGDB_C012151
PGDB_AS000508
View
DC50
-
=
47.6
nM
-
—
WIZ
-
HT-1080
WO2025256460A1
PGDB_A011316
PGDB_C012156
PGDB_AS000508
View
DC50
-
=
121
nM
-
—
WIZ
-
HT-1080
WO2025256460A1
PGDB_A011376
PGDB_C012147
PGDB_AS000508
View
DC50
-
=
10.7
nM
-
—
WIZ
-
HT-1080
WO2025256460A1
PGDB_A012645
PGDB_C012094
PGDB_AS000508
View
DC50
-
=
47.8
nM
-
—
WIZ
-
HT-1080
WO2025256460A1
PGDB_A012833
PGDB_C012052
PGDB_AS000508
View
DC50
-
=
118
nM
-
—
WIZ
-
HT-1080
WO2025256460A1
PGDB_A013540
PGDB_C012078
PGDB_AS000508
View
DC50
-
=
33.3
nM
-
—
WIZ
-
HT-1080
WO2025256460A1
PGDB_A014052
PGDB_C012082
PGDB_AS000508
View
DC50
-
=
130
nM
-
—
WIZ
-
HT-1080
WO2025256460A1
PGDB_A014975
PGDB_C012063
PGDB_AS000508
View
DC50
-
=
47.8
nM
-
—
WIZ
-
HT-1080
WO2025256460A1
PGDB_A015206
PGDB_C012122
PGDB_AS000508
View
DC50
-
=
22.6
nM
-
—
WIZ
-
HT-1080
WO2025256460A1
PGDB_A015242
PGDB_C012095
PGDB_AS000508
View
DC50
-
=
11
nM
-
—
WIZ
-
HT-1080
WO2025256460A1
PGDB_A015395
PGDB_C012135
PGDB_AS000508
View
DC50
-
=
112
nM
-
—
WIZ
-
HT-1080
WO2025256460A1
PGDB_A015922
PGDB_C012049
PGDB_AS000508
View
DC50
-
=
127
nM
-
—
WIZ
-
HT-1080
WO2025256460A1
PGDB_A016492
PGDB_C012083
PGDB_AS000508
View
DC50
-
=
130
nM
-
—
WIZ
-
HT-1080
WO2025256460A1
PGDB_A016750
PGDB_C012076
PGDB_AS000508
View