Assay context summary

Assay context

36 activity records
Activity compounds and values

Activity records

36 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C031974
IC50-=4.5nM--CRBNSW1990WO2026114958A1PGDB_A001661PGDB_C031974PGDB_AS000509View
2D structure for PGDB_C031995
IC50-=9.2nM--CRBNSW1990WO2026114958A1PGDB_A002482PGDB_C031995PGDB_AS000509View
2D structure for PGDB_C031972
IC50-=14.3nM--CRBNSW1990WO2026114958A1PGDB_A002812PGDB_C031972PGDB_AS000509View
2D structure for PGDB_C031946
IC50-=171.5nM--CRBNSW1990WO2026114958A1PGDB_A002963PGDB_C031946PGDB_AS000509View
2D structure for PGDB_C031975
IC50-=13.6nM--CRBNSW1990WO2026114958A1PGDB_A002965PGDB_C031975PGDB_AS000509View
2D structure for PGDB_C031970
IC50-=46.8nM--CRBNSW1990WO2026114958A1PGDB_A003006PGDB_C031970PGDB_AS000509View
2D structure for PGDB_C031967
IC50-=15.1nM--CRBNSW1990WO2026114958A1PGDB_A003093PGDB_C031967PGDB_AS000509View
2D structure for PGDB_C031952
IC50-=22.2nM--CRBNSW1990WO2026114958A1PGDB_A003147PGDB_C031952PGDB_AS000509View
2D structure for PGDB_C031993
IC50-=19.2nM--CRBNSW1990WO2026114958A1PGDB_A003224PGDB_C031993PGDB_AS000509View
2D structure for PGDB_C031968
IC50-=6.8nM--CRBNSW1990WO2026114958A1PGDB_A003974PGDB_C031968PGDB_AS000509View
2D structure for PGDB_C031973
IC50-=21.5nM--CRBNSW1990WO2026114958A1PGDB_A004219PGDB_C031973PGDB_AS000509View
2D structure for PGDB_C031991
IC50-=24.3nM--CRBNSW1990WO2026114958A1PGDB_A004273PGDB_C031991PGDB_AS000509View
2D structure for PGDB_C031954
IC50-=76.5nM--CRBNSW1990WO2026114958A1PGDB_A004302PGDB_C031954PGDB_AS000509View
2D structure for PGDB_C031988
IC50-=1000nM--CRBNSW1990WO2026114958A1PGDB_A004598PGDB_C031988PGDB_AS000509View
2D structure for PGDB_C031971
IC50-=10.4nM--CRBNSW1990WO2026114958A1PGDB_A004805PGDB_C031971PGDB_AS000509View
2D structure for PGDB_C031969
IC50-=12.3nM--CRBNSW1990WO2026114958A1PGDB_A005229PGDB_C031969PGDB_AS000509View
2D structure for PGDB_C031941
IC50-=2.6nM--CRBNSW1990WO2026114958A1PGDB_A005283PGDB_C031941PGDB_AS000509View
2D structure for PGDB_C031976
IC50-=57.3nM--CRBNSW1990WO2026114958A1PGDB_A005300PGDB_C031976PGDB_AS000509View
2D structure for PGDB_C031947
IC50-=70.9nM--CRBNSW1990WO2026114958A1PGDB_A006179PGDB_C031947PGDB_AS000509View
2D structure for PGDB_C031960
IC50-=12.6nM--CRBNSW1990WO2026114958A1PGDB_A006183PGDB_C031960PGDB_AS000509View