Assay
PGDB_AS000540
System: cell_basedCell line: Mino
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 50-100 | nM | - | — | BTK | CRBN | Mino | CN116239566A | PGDB_A009559 | PGDB_C025814 | PGDB_AS000540 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | CRBN | Mino | CN116239566A | PGDB_A018292 | PGDB_C019593 | PGDB_AS000540 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | CRBN | Mino | CN116239566A | PGDB_A024648 | PGDB_C025803 | PGDB_AS000540 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | CRBN | Mino | CN116239566A | PGDB_A054274 | PGDB_C025807 | PGDB_AS000540 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | CRBN | Mino | CN116239566A | PGDB_A062364 | PGDB_C015982 | PGDB_AS000540 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | CRBN | Mino | CN116239566A | PGDB_A068632 | PGDB_C025815 | PGDB_AS000540 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | CRBN | Mino | CN116239566A | PGDB_A077649 | PGDB_C025809 | PGDB_AS000540 | View |