Assay
PGDB_AS000559
System: cell_basedCell line: H1975
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 50-100 | nM | - | — | - | - | H1975 | WO2025016359A1 | PGDB_A015486 | PGDB_C019358 | PGDB_AS000559 | View | |
| IC50 | - | = | 1-5 | nM | - | — | - | - | H1975 | WO2025016359A1 | PGDB_A033389 | PGDB_C019354 | PGDB_AS000559 | View | |
| IC50 | - | = | 1-5 | nM | - | — | - | - | H1975 | WO2025016359A1 | PGDB_A037419 | PGDB_C019344 | PGDB_AS000559 | View | |
| IC50 | - | = | 50-100 | nM | - | — | - | - | H1975 | WO2025016359A1 | PGDB_A038302 | PGDB_C019363 | PGDB_AS000559 | View | |
| IC50 | - | = | 1-5 | nM | - | — | - | - | H1975 | WO2025016359A1 | PGDB_A053535 | PGDB_C019371 | PGDB_AS000559 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | - | - | H1975 | WO2025016359A1 | PGDB_A054528 | PGDB_C019374 | PGDB_AS000559 | View | |
| IC50 | - | = | 100-500 | nM | - | — | - | - | H1975 | WO2025016359A1 | PGDB_A057077 | PGDB_C019469 | PGDB_AS000559 | View | |
| IC50 | - | = | 1-5 | nM | - | — | - | - | H1975 | WO2025016359A1 | PGDB_A060623 | PGDB_C019364 | PGDB_AS000559 | View | |
| IC50 | - | = | 100-500 | nM | - | — | - | - | H1975 | WO2025016359A1 | PGDB_A068985 | PGDB_C019352 | PGDB_AS000559 | View | |
| IC50 | - | = | 50-100 | nM | - | — | - | - | H1975 | WO2025016359A1 | PGDB_A077253 | PGDB_C019342 | PGDB_AS000559 | View |