Assay context summary

Assay context

32 activity records
Activity compounds and values

Activity records

32 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C005479
IC50-=14.99nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A009609PGDB_C005479PGDB_AS000582View
2D structure for PGDB_C005496
IC50-=14.06nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A010402PGDB_C005496PGDB_AS000582View
2D structure for PGDB_C005502
IC50-=40.39nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A010559PGDB_C005502PGDB_AS000582View
2D structure for PGDB_C003382
IC50-=62.69nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A010893PGDB_C003382PGDB_AS000582View
2D structure for PGDB_C005486
IC50-=11.36nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A016912PGDB_C005486PGDB_AS000582View
2D structure for PGDB_C005478
IC50-=10.08nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A017687PGDB_C005478PGDB_AS000582View
2D structure for PGDB_C005501
IC50-=90.69nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A017968PGDB_C005501PGDB_AS000582View
2D structure for PGDB_C005481
IC50-=58.39nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A018407PGDB_C005481PGDB_AS000582View
2D structure for PGDB_C005490
IC50-=23.11nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A021436PGDB_C005490PGDB_AS000582View
2D structure for PGDB_C005497
IC50-=13.91nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A024792PGDB_C005497PGDB_AS000582View
2D structure for PGDB_C005506
IC50-=18.43nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A032172PGDB_C005506PGDB_AS000582View
2D structure for PGDB_C005494
IC50-=13.31nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A032450PGDB_C005494PGDB_AS000582View
2D structure for PGDB_C005485
IC50-=10.31nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A037279PGDB_C005485PGDB_AS000582View
2D structure for PGDB_C005489
IC50-=20.32nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A037610PGDB_C005489PGDB_AS000582View
2D structure for PGDB_C005500
IC50-=24.67nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A038043PGDB_C005500PGDB_AS000582View
2D structure for PGDB_C005488
IC50-=9.3nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A038548PGDB_C005488PGDB_AS000582View
2D structure for PGDB_C005498
IC50-=40.86nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A040429PGDB_C005498PGDB_AS000582View
2D structure for PGDB_C005505
IC50-=33.37nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A040731PGDB_C005505PGDB_AS000582View
2D structure for PGDB_C005482
IC50-=22.71nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A046330PGDB_C005482PGDB_AS000582View
2D structure for PGDB_C005484
IC50-=22.59nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A046782PGDB_C005484PGDB_AS000582View