Assay context summary

Assay context

20 activity records
Activity compounds and values

Activity records

20 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C001841
IC50-=0.06uM-CSNK1A1-MV-4-11WO2022257897A1PGDB_A007363PGDB_C001841PGDB_AS000623View
2D structure for PGDB_C001833
IC50-=0.128uM-CSNK1A1-MV-4-11WO2022257897A1PGDB_A018574PGDB_C001833PGDB_AS000623View
2D structure for PGDB_C001808
IC50-=0.42uM-CSNK1A1-MV-4-11WO2022257897A1PGDB_A020001PGDB_C001808PGDB_AS000623View
2D structure for PGDB_C001860
IC50-=0.102uM-CSNK1A1-MV-4-11WO2022257897A1PGDB_A021969PGDB_C001860PGDB_AS000623View
2D structure for PGDB_C001858
IC50-=0.071uM-CSNK1A1-MV-4-11WO2022257897A1PGDB_A026352PGDB_C001858PGDB_AS000623View
2D structure for PGDB_C001786
IC50-=0.198uM-CSNK1A1-MV-4-11WO2022257897A1PGDB_A027823PGDB_C001786PGDB_AS000623View
2D structure for PGDB_C001864
IC50-=0.198uM-CSNK1A1-MV-4-11WO2022257897A1PGDB_A028562PGDB_C001864PGDB_AS000623View
2D structure for PGDB_C001859
IC50-=0.024uM-CSNK1A1-MV-4-11WO2022257897A1PGDB_A030053PGDB_C001859PGDB_AS000623View
2D structure for PGDB_C001842
IC50-=0.027uM-CSNK1A1-MV-4-11WO2022257897A1PGDB_A034190PGDB_C001842PGDB_AS000623View
2D structure for PGDB_C001791
IC50-=0.691uM-CSNK1A1-MV-4-11WO2022257897A1PGDB_A035024PGDB_C001791PGDB_AS000623View
2D structure for PGDB_C001837
IC50-=0.176uM-CSNK1A1-MV-4-11WO2022257897A1PGDB_A035378PGDB_C001837PGDB_AS000623View
2D structure for PGDB_C001861
IC50-=0.142uM-CSNK1A1-MV-4-11WO2022257897A1PGDB_A036842PGDB_C001861PGDB_AS000623View
2D structure for PGDB_C001785
IC50-=0.262uM-CSNK1A1-MV-4-11WO2022257897A1PGDB_A039020PGDB_C001785PGDB_AS000623View
2D structure for PGDB_C001807
IC50-=0.115uM-CSNK1A1-MV-4-11WO2022257897A1PGDB_A040004PGDB_C001807PGDB_AS000623View
2D structure for PGDB_C001862
IC50-=0.133uM-CSNK1A1-MV-4-11WO2022257897A1PGDB_A044384PGDB_C001862PGDB_AS000623View
2D structure for PGDB_C001792
IC50-=0.205uM-CSNK1A1-MV-4-11WO2022257897A1PGDB_A048325PGDB_C001792PGDB_AS000623View
2D structure for PGDB_C001793
IC50-=0.172uM-CSNK1A1-MV-4-11WO2022257897A1PGDB_A063800PGDB_C001793PGDB_AS000623View
2D structure for PGDB_C001838
IC50-=0.176uM-CSNK1A1-MV-4-11WO2022257897A1PGDB_A068339PGDB_C001838PGDB_AS000623View
2D structure for PGDB_C001784
IC50-=0.112uM-CSNK1A1-MV-4-11WO2022257897A1PGDB_A075950PGDB_C001784PGDB_AS000623View
2D structure for PGDB_C001790
IC50-=0.363uM-CSNK1A1-MV-4-11WO2022257897A1PGDB_A076133PGDB_C001790PGDB_AS000623View