Assay context summary

Assay context

130 activity records
Activity compounds and values

Activity records

130 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C031257
DC50-=17nM-NEK7-CAL-51WO2026099466A1PGDB_A000222PGDB_C031257PGDB_AS000897View
2D structure for PGDB_C031208
DC50-=159nM-NEK7-CAL-51WO2026099466A1PGDB_A000371PGDB_C031208PGDB_AS000897View
2D structure for PGDB_C031239
DC50-=79nM-NEK7-CAL-51WO2026099466A1PGDB_A000405PGDB_C031239PGDB_AS000897View
2D structure for PGDB_C031273
DC50-=8nM-NEK7-CAL-51WO2026099466A1PGDB_A000457PGDB_C031273PGDB_AS000897View
2D structure for PGDB_C031272
DC50-=183nM-NEK7-CAL-51WO2026099466A1PGDB_A000745PGDB_C031272PGDB_AS000897View
2D structure for PGDB_C031290
DC50-=46nM-NEK7-CAL-51WO2026099466A1PGDB_A000866PGDB_C031290PGDB_AS000897View
2D structure for PGDB_C031221
DC50-=50nM-NEK7-CAL-51WO2026099466A1PGDB_A000876PGDB_C031221PGDB_AS000897View
2D structure for PGDB_C031280
DC50-=107nM-NEK7-CAL-51WO2026099466A1PGDB_A000938PGDB_C031280PGDB_AS000897View
2D structure for PGDB_C031247
DC50-=56nM-NEK7-CAL-51WO2026099466A1PGDB_A000979PGDB_C031247PGDB_AS000897View
2D structure for PGDB_C031256
DC50-=112nM-NEK7-CAL-51WO2026099466A1PGDB_A001033PGDB_C031256PGDB_AS000897View
2D structure for PGDB_C031212
DC50-=2nM-NEK7-CAL-51WO2026099466A1PGDB_A001059PGDB_C031212PGDB_AS000897View
2D structure for PGDB_C031244
DC50-=104nM-NEK7-CAL-51WO2026099466A1PGDB_A001228PGDB_C031244PGDB_AS000897View
2D structure for PGDB_C031253
DC50-=126nM-NEK7-CAL-51WO2026099466A1PGDB_A001300PGDB_C031253PGDB_AS000897View
2D structure for PGDB_C031213
DC50-=70nM-NEK7-CAL-51WO2026099466A1PGDB_A001345PGDB_C031213PGDB_AS000897View
2D structure for PGDB_C031224
DC50-=50nM-NEK7-CAL-51WO2026099466A1PGDB_A001369PGDB_C031224PGDB_AS000897View
2D structure for PGDB_C031270
DC50-=190nM-NEK7-CAL-51WO2026099466A1PGDB_A001398PGDB_C031270PGDB_AS000897View
2D structure for PGDB_C031269
DC50-=37nM-NEK7-CAL-51WO2026099466A1PGDB_A001441PGDB_C031269PGDB_AS000897View
2D structure for PGDB_C031274
DC50-=25nM-NEK7-CAL-51WO2026099466A1PGDB_A001483PGDB_C031274PGDB_AS000897View
2D structure for PGDB_C031323
DC50-=304nM-NEK7-CAL-51WO2026099466A1PGDB_A001806PGDB_C031323PGDB_AS000897View
2D structure for PGDB_C031260
DC50-=129nM-NEK7-CAL-51WO2026099466A1PGDB_A001842PGDB_C031260PGDB_AS000897View