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SIMM · NJU
Assay
PGDB_AS000897
System: cell_based
Target: NEK7
Cell line: CAL-51
Assay context summary
Assay context
130 activity records
Assay family
% Degradation
System
cell_based
Readout
DC50
Target
NEK7
E3
Not specified
Cell line
CAL-51
Organism
Homo sapiens
Technology
luminescence
Activity compounds and values
Activity records
130 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
DC50
-
=
17
nM
-
—
NEK7
-
CAL-51
WO2026099466A1
PGDB_A000222
PGDB_C031257
PGDB_AS000897
View
DC50
-
=
159
nM
-
—
NEK7
-
CAL-51
WO2026099466A1
PGDB_A000371
PGDB_C031208
PGDB_AS000897
View
DC50
-
=
79
nM
-
—
NEK7
-
CAL-51
WO2026099466A1
PGDB_A000405
PGDB_C031239
PGDB_AS000897
View
DC50
-
=
8
nM
-
—
NEK7
-
CAL-51
WO2026099466A1
PGDB_A000457
PGDB_C031273
PGDB_AS000897
View
DC50
-
=
183
nM
-
—
NEK7
-
CAL-51
WO2026099466A1
PGDB_A000745
PGDB_C031272
PGDB_AS000897
View
DC50
-
=
46
nM
-
—
NEK7
-
CAL-51
WO2026099466A1
PGDB_A000866
PGDB_C031290
PGDB_AS000897
View
DC50
-
=
50
nM
-
—
NEK7
-
CAL-51
WO2026099466A1
PGDB_A000876
PGDB_C031221
PGDB_AS000897
View
DC50
-
=
107
nM
-
—
NEK7
-
CAL-51
WO2026099466A1
PGDB_A000938
PGDB_C031280
PGDB_AS000897
View
DC50
-
=
56
nM
-
—
NEK7
-
CAL-51
WO2026099466A1
PGDB_A000979
PGDB_C031247
PGDB_AS000897
View
DC50
-
=
112
nM
-
—
NEK7
-
CAL-51
WO2026099466A1
PGDB_A001033
PGDB_C031256
PGDB_AS000897
View
DC50
-
=
2
nM
-
—
NEK7
-
CAL-51
WO2026099466A1
PGDB_A001059
PGDB_C031212
PGDB_AS000897
View
DC50
-
=
104
nM
-
—
NEK7
-
CAL-51
WO2026099466A1
PGDB_A001228
PGDB_C031244
PGDB_AS000897
View
DC50
-
=
126
nM
-
—
NEK7
-
CAL-51
WO2026099466A1
PGDB_A001300
PGDB_C031253
PGDB_AS000897
View
DC50
-
=
70
nM
-
—
NEK7
-
CAL-51
WO2026099466A1
PGDB_A001345
PGDB_C031213
PGDB_AS000897
View
DC50
-
=
50
nM
-
—
NEK7
-
CAL-51
WO2026099466A1
PGDB_A001369
PGDB_C031224
PGDB_AS000897
View
DC50
-
=
190
nM
-
—
NEK7
-
CAL-51
WO2026099466A1
PGDB_A001398
PGDB_C031270
PGDB_AS000897
View
DC50
-
=
37
nM
-
—
NEK7
-
CAL-51
WO2026099466A1
PGDB_A001441
PGDB_C031269
PGDB_AS000897
View
DC50
-
=
25
nM
-
—
NEK7
-
CAL-51
WO2026099466A1
PGDB_A001483
PGDB_C031274
PGDB_AS000897
View
DC50
-
=
304
nM
-
—
NEK7
-
CAL-51
WO2026099466A1
PGDB_A001806
PGDB_C031323
PGDB_AS000897
View
DC50
-
=
129
nM
-
—
NEK7
-
CAL-51
WO2026099466A1
PGDB_A001842
PGDB_C031260
PGDB_AS000897
View