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SIMM · NJU
Assay
PGDB_AS000941
System: cell_based
Cell line: REC-1
Assay context summary
Assay context
70 activity records
Assay family
viability
System
cell_based
Readout
IC50
E3
Not specified
Cell line
REC-1
Organism
Homo sapiens
Technology
luminescence
Detection target
% Cell viability
Activity compounds and values
Activity records
70 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
IC50
-
=
87.83
nM
-
—
VAV1
-
REC-1
WO2026103798A1
PGDB_A000030
PGDB_C031353
PGDB_AS000941
View
IC50
-
=
161.56
nM
-
—
VAV1
-
REC-1
WO2026103798A1
PGDB_A000041
PGDB_C031339
PGDB_AS000941
View
IC50
-
=
15.8
nM
-
—
VAV1
-
REC-1
WO2026103798A1
PGDB_A000383
PGDB_C031376
PGDB_AS000941
View
IC50
-
=
563.56
nM
-
—
VAV1
-
REC-1
WO2026103798A1
PGDB_A000658
PGDB_C031388
PGDB_AS000941
View
IC50
-
=
1.99
nM
-
—
VAV1
-
REC-1
WO2026103798A1
PGDB_A000686
PGDB_C031357
PGDB_AS000941
View
IC50
-
=
42.77
nM
-
—
VAV1
-
REC-1
WO2026103798A1
PGDB_A000707
PGDB_C031354
PGDB_AS000941
View
IC50
-
=
16.47
nM
-
—
VAV1
-
REC-1
WO2026103798A1
PGDB_A000969
PGDB_C031380
PGDB_AS000941
View
IC50
-
=
244
nM
-
—
VAV1
-
REC-1
WO2026103798A1
PGDB_A001063
PGDB_C031340
PGDB_AS000941
View
IC50
-
=
1.95
nM
-
—
VAV1
-
REC-1
WO2026103798A1
PGDB_A001610
PGDB_C031342
PGDB_AS000941
View
IC50
-
=
19.82
nM
-
—
VAV1
-
REC-1
WO2026103798A1
PGDB_A001807
PGDB_C031374
PGDB_AS000941
View
IC50
-
=
196.45
nM
-
—
VAV1
-
REC-1
WO2026103798A1
PGDB_A002101
PGDB_C031386
PGDB_AS000941
View
IC50
-
=
6.92
nM
-
—
VAV1
-
REC-1
WO2026103798A1
PGDB_A002265
PGDB_C031379
PGDB_AS000941
View
IC50
-
=
24.78
nM
-
—
VAV1
-
REC-1
WO2026103798A1
PGDB_A002433
PGDB_C031345
PGDB_AS000941
View
IC50
-
=
2.21
nM
-
—
VAV1
-
REC-1
WO2026103798A1
PGDB_A002575
PGDB_C031365
PGDB_AS000941
View
IC50
-
=
33.85
nM
-
—
VAV1
-
REC-1
WO2026103798A1
PGDB_A002723
PGDB_C031369
PGDB_AS000941
View
IC50
-
=
2.26
nM
-
—
VAV1
-
REC-1
WO2026103798A1
PGDB_A002727
PGDB_C031356
PGDB_AS000941
View
IC50
-
=
14.39
nM
-
—
VAV1
-
REC-1
WO2026103798A1
PGDB_A002861
PGDB_C031390
PGDB_AS000941
View
IC50
-
=
31.41
nM
-
—
VAV1
-
REC-1
WO2026103798A1
PGDB_A002994
PGDB_C031335
PGDB_AS000941
View
IC50
-
=
104.49
nM
-
—
VAV1
-
REC-1
WO2026103798A1
PGDB_A003145
PGDB_C031392
PGDB_AS000941
View
IC50
-
=
31.66
nM
-
—
VAV1
-
REC-1
WO2026103798A1
PGDB_A003202
PGDB_C031384
PGDB_AS000941
View