Assay context summary

Assay context

70 activity records
Activity compounds and values

Activity records

70 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C031353
IC50-=87.83nM-VAV1-REC-1WO2026103798A1PGDB_A000030PGDB_C031353PGDB_AS000941View
2D structure for PGDB_C031339
IC50-=161.56nM-VAV1-REC-1WO2026103798A1PGDB_A000041PGDB_C031339PGDB_AS000941View
2D structure for PGDB_C031376
IC50-=15.8nM-VAV1-REC-1WO2026103798A1PGDB_A000383PGDB_C031376PGDB_AS000941View
2D structure for PGDB_C031388
IC50-=563.56nM-VAV1-REC-1WO2026103798A1PGDB_A000658PGDB_C031388PGDB_AS000941View
2D structure for PGDB_C031357
IC50-=1.99nM-VAV1-REC-1WO2026103798A1PGDB_A000686PGDB_C031357PGDB_AS000941View
2D structure for PGDB_C031354
IC50-=42.77nM-VAV1-REC-1WO2026103798A1PGDB_A000707PGDB_C031354PGDB_AS000941View
2D structure for PGDB_C031380
IC50-=16.47nM-VAV1-REC-1WO2026103798A1PGDB_A000969PGDB_C031380PGDB_AS000941View
2D structure for PGDB_C031340
IC50-=244nM-VAV1-REC-1WO2026103798A1PGDB_A001063PGDB_C031340PGDB_AS000941View
2D structure for PGDB_C031342
IC50-=1.95nM-VAV1-REC-1WO2026103798A1PGDB_A001610PGDB_C031342PGDB_AS000941View
2D structure for PGDB_C031374
IC50-=19.82nM-VAV1-REC-1WO2026103798A1PGDB_A001807PGDB_C031374PGDB_AS000941View
2D structure for PGDB_C031386
IC50-=196.45nM-VAV1-REC-1WO2026103798A1PGDB_A002101PGDB_C031386PGDB_AS000941View
2D structure for PGDB_C031379
IC50-=6.92nM-VAV1-REC-1WO2026103798A1PGDB_A002265PGDB_C031379PGDB_AS000941View
2D structure for PGDB_C031345
IC50-=24.78nM-VAV1-REC-1WO2026103798A1PGDB_A002433PGDB_C031345PGDB_AS000941View
2D structure for PGDB_C031365
IC50-=2.21nM-VAV1-REC-1WO2026103798A1PGDB_A002575PGDB_C031365PGDB_AS000941View
2D structure for PGDB_C031369
IC50-=33.85nM-VAV1-REC-1WO2026103798A1PGDB_A002723PGDB_C031369PGDB_AS000941View
2D structure for PGDB_C031356
IC50-=2.26nM-VAV1-REC-1WO2026103798A1PGDB_A002727PGDB_C031356PGDB_AS000941View
2D structure for PGDB_C031390
IC50-=14.39nM-VAV1-REC-1WO2026103798A1PGDB_A002861PGDB_C031390PGDB_AS000941View
2D structure for PGDB_C031335
IC50-=31.41nM-VAV1-REC-1WO2026103798A1PGDB_A002994PGDB_C031335PGDB_AS000941View
2D structure for PGDB_C031392
IC50-=104.49nM-VAV1-REC-1WO2026103798A1PGDB_A003145PGDB_C031392PGDB_AS000941View
2D structure for PGDB_C031384
IC50-=31.66nM-VAV1-REC-1WO2026103798A1PGDB_A003202PGDB_C031384PGDB_AS000941View