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Compound
PGDB_C031356
4 activity records1 related patents
2D structure
[2H]C1([2H])CC([2H])([2H])N(C2(C)CC2)C(=O)N1c1ccc(-c2cccc(C3CCC(=O)NC3=O)c2Cl)cc1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | = | 0.81 | nM | - | — | VAV1 | - | REC-1 | WO2026103798A1 | PGDB_A002494 | PGDB_C031356 | PGDB_AS000225 | View |
| IC50 | - | = | 2.26 | nM | - | — | VAV1 | - | REC-1 | WO2026103798A1 | PGDB_A002727 | PGDB_C031356 | PGDB_AS000941 | View |
| DC50 | - | <= | 100 | nM | - | — | VAV1 | - | REC-1 | WO2026103798A1 | PGDB_A004327 | PGDB_C031356 | PGDB_AS002449 | View |
| Fold change | 185 | = | 0.29 | fold | - | 72 h | VAV1 | - | - | WO2026103798A1 | PGDB_A078462 | PGDB_C031356 | PGDB_AS001694 | View |