Assay

PGDB_AS001045

System: cell_basedTarget: KRAS
Assay context summary

Assay context

57 activity records
Assay family% Degradation
Systemcell_based
ReadoutDC50
TargetKRAS
E3Not specified
OrganismHomo sapiens
Technologyluminescence
Activity compounds and values

Activity records

57 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C031972
DC50-=2nM-—KRAS--WO2026114958A1PGDB_A000262PGDB_C031972PGDB_AS001045View
2D structure for PGDB_C031947
DC50-=3.1nM-—KRAS--WO2026114958A1PGDB_A000381PGDB_C031947PGDB_AS001045View
2D structure for PGDB_C031991
DC50-=1.4nM-—KRAS--WO2026114958A1PGDB_A000388PGDB_C031991PGDB_AS001045View
2D structure for PGDB_C031984
DC50-=2.7nM-—KRAS--WO2026114958A1PGDB_A000523PGDB_C031984PGDB_AS001045View
2D structure for PGDB_C031966
DC50-=14nM-—KRAS--WO2026114958A1PGDB_A000727PGDB_C031966PGDB_AS001045View
2D structure for PGDB_C031946
DC50-=2.4nM-—KRAS--WO2026114958A1PGDB_A000779PGDB_C031946PGDB_AS001045View
2D structure for PGDB_C031992
DC50-=4.8nM-—KRAS--WO2026114958A1PGDB_A000842PGDB_C031992PGDB_AS001045View
2D structure for PGDB_C031976
DC50-=9.4nM-—KRAS--WO2026114958A1PGDB_A000984PGDB_C031976PGDB_AS001045View
2D structure for PGDB_C031959
DC50-=4nM-—KRAS--WO2026114958A1PGDB_A001145PGDB_C031959PGDB_AS001045View
2D structure for PGDB_C031953
DC50-=2.7nM-—KRAS--WO2026114958A1PGDB_A001221PGDB_C031953PGDB_AS001045View
2D structure for PGDB_C031975
DC50-=3.1nM-—KRAS--WO2026114958A1PGDB_A001560PGDB_C031975PGDB_AS001045View
2D structure for PGDB_C031973
DC50-=1.9nM-—KRAS--WO2026114958A1PGDB_A001683PGDB_C031973PGDB_AS001045View
2D structure for PGDB_C031978
DC50-=2.8nM-—KRAS--WO2026114958A1PGDB_A001921PGDB_C031978PGDB_AS001045View
2D structure for PGDB_C031981
DC50-=3.6nM-—KRAS--WO2026114958A1PGDB_A001941PGDB_C031981PGDB_AS001045View
2D structure for PGDB_C031994
DC50-=0.7nM-—KRAS--WO2026114958A1PGDB_A002026PGDB_C031994PGDB_AS001045View
2D structure for PGDB_C031974
DC50-=2.7nM-—KRAS--WO2026114958A1PGDB_A002077PGDB_C031974PGDB_AS001045View
2D structure for PGDB_C031982
DC50-=3.2nM-—KRAS--WO2026114958A1PGDB_A002127PGDB_C031982PGDB_AS001045View
2D structure for PGDB_C031979
DC50-=9nM-—KRAS--WO2026114958A1PGDB_A002508PGDB_C031979PGDB_AS001045View
2D structure for PGDB_C031965
DC50-=1.5nM-—KRAS--WO2026114958A1PGDB_A002523PGDB_C031965PGDB_AS001045View
2D structure for PGDB_C031967
DC50-=3.4nM-—KRAS--WO2026114958A1PGDB_A002906PGDB_C031967PGDB_AS001045View
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