Assay context summary

Assay context

379 activity records
Activity compounds and values

Activity records

379 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C020068
% Degradation->=20%Concentration series: 500 nM, 50 nM24 hGSPT1--WO2024245444A1PGDB_A007105PGDB_C020068PGDB_AS001137View
2D structure for PGDB_C020059
% Degradation-<20%Concentration series: 500 nM, 50 nM24 hGSPT1--WO2024245444A1PGDB_A007353PGDB_C020059PGDB_AS001137View
2D structure for PGDB_C014248
% Degradation->=20%Concentration series: 500 nM, 50 nM24 hGSPT1--WO2024245444A1PGDB_A007435PGDB_C014248PGDB_AS001137View
2D structure for PGDB_C020066
% Degradation-<20%Concentration series: 500 nM, 50 nM24 hGSPT1--WO2024245444A1PGDB_A007472PGDB_C020066PGDB_AS001137View
2D structure for PGDB_C020165
% Degradation->=20%Concentration series: 500 nM, 50 nM24 hGSPT1--WO2024245444A1PGDB_A007650PGDB_C020165PGDB_AS001137View
2D structure for PGDB_C020103
% Degradation->=20%Concentration series: 500 nM, 50 nM24 hGSPT1--WO2024245444A1PGDB_A007863PGDB_C020103PGDB_AS001137View
2D structure for PGDB_C020129
% Degradation->=20%Concentration series: 500 nM, 50 nM24 hGSPT1--WO2024245444A1PGDB_A008538PGDB_C020129PGDB_AS001137View
2D structure for PGDB_C014298
% Degradation->=20%Concentration series: 500 nM, 50 nM24 hGSPT1--WO2024245444A1PGDB_A009041PGDB_C014298PGDB_AS001137View
2D structure for PGDB_C020123
% Degradation->=20%Concentration series: 500 nM, 50 nM24 hGSPT1--WO2024245444A1PGDB_A009176PGDB_C020123PGDB_AS001137View
2D structure for PGDB_C020122
% Degradation->=20%Concentration series: 500 nM, 50 nM24 hGSPT1--WO2024245444A1PGDB_A009216PGDB_C020122PGDB_AS001137View
2D structure for PGDB_C014310
% Degradation->=20%Concentration series: 500 nM, 50 nM24 hGSPT1--WO2024245444A1PGDB_A009239PGDB_C014310PGDB_AS001137View
2D structure for PGDB_C019986
% Degradation-<20%Concentration series: 500 nM, 50 nM24 hGSPT1--WO2024245444A1PGDB_A009555PGDB_C019986PGDB_AS001137View
2D structure for PGDB_C020092
% Degradation->=20%Concentration series: 500 nM, 50 nM24 hGSPT1--WO2024245444A1PGDB_A009625PGDB_C020092PGDB_AS001137View
2D structure for PGDB_C020167
% Degradation->=20%Concentration series: 500 nM, 50 nM24 hGSPT1--WO2024245444A1PGDB_A009642PGDB_C020167PGDB_AS001137View
2D structure for PGDB_C020056
% Degradation->=20%Concentration series: 500 nM, 50 nM24 hGSPT1--WO2024245444A1PGDB_A009914PGDB_C020056PGDB_AS001137View
2D structure for PGDB_C019953
% Degradation->=20%Concentration series: 500 nM, 50 nM24 hGSPT1--WO2024245444A1PGDB_A009991PGDB_C019953PGDB_AS001137View
2D structure for PGDB_C014241
% Degradation->=20%Concentration series: 500 nM, 50 nM24 hGSPT1--WO2024245444A1PGDB_A010374PGDB_C014241PGDB_AS001137View
2D structure for PGDB_C020000
% Degradation-<20%Concentration series: 500 nM, 50 nM24 hGSPT1--WO2024245444A1PGDB_A010377PGDB_C020000PGDB_AS001137View
2D structure for PGDB_C020047
% Degradation-<20%Concentration series: 500 nM, 50 nM24 hGSPT1--WO2024245444A1PGDB_A010427PGDB_C020047PGDB_AS001137View
2D structure for PGDB_C014257
% Degradation->=20%Concentration series: 500 nM, 50 nM24 hGSPT1--WO2024245444A1PGDB_A010765PGDB_C014257PGDB_AS001137View