Assay

PGDB_AS001164

System: cell_basedTarget: GSPT1Cell line: 293A
Assay context summary

Assay context

10 activity records
Assay family% Degradation
Systemcell_based
ReadoutDC50
TargetGSPT1
E3Not specified
Cell line293A
Detection targetprotein_degradation
Activity compounds and values

Activity records

10 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C001073
DC50->5uM-—GSPT1-293ACN121591645APGDB_A007067PGDB_C001073PGDB_AS001164View
2D structure for PGDB_C001070
DC50-=0.522uM-—GSPT1-293ACN121591645APGDB_A012411PGDB_C001070PGDB_AS001164View
2D structure for PGDB_C001079
DC50-=0.0193uM-—GSPT1-293ACN121591645APGDB_A014521PGDB_C001079PGDB_AS001164View
2D structure for PGDB_C001078
DC50->5uM-—GSPT1-293ACN121591645APGDB_A021362PGDB_C001078PGDB_AS001164View
2D structure for PGDB_C001075
DC50-=0.00277uM-—GSPT1-293ACN121591645APGDB_A024601PGDB_C001075PGDB_AS001164View
2D structure for PGDB_C001077
DC50-=0.0695uM-—GSPT1-293ACN121591645APGDB_A028248PGDB_C001077PGDB_AS001164View
2D structure for PGDB_C001074
DC50-=0.067uM-—GSPT1-293ACN121591645APGDB_A043447PGDB_C001074PGDB_AS001164View
2D structure for PGDB_C001076
DC50->5uM-—GSPT1-293ACN121591645APGDB_A043508PGDB_C001076PGDB_AS001164View
2D structure for PGDB_C001072
DC50-=0.00167uM-—GSPT1-293ACN121591645APGDB_A070065PGDB_C001072PGDB_AS001164View
2D structure for PGDB_C001071
DC50-=0.00196uM-—GSPT1-293ACN121591645APGDB_A071384PGDB_C001071PGDB_AS001164View
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