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SIMM · NJU
Assay
PGDB_AS001212
System: cell_based
Target: GSPT1
Cell line: HL-60
Assay context summary
Assay context
36 activity records
Assay family
% Degradation
System
cell_based
Readout
percent_remaining
Target
GSPT1
E3
Not specified
Cell line
HL-60
Technology
Western_blot
Activity compounds and values
Activity records
36 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
% Degradation
-
=
95
%
10 nM
24 h
-
-
HL-60
CN117982498A
PGDB_A011941
PGDB_C000556
PGDB_AS001212
View
% Degradation
-
=
100
%
10 nM
24 h
-
-
HL-60
CN117982498A
PGDB_A014243
PGDB_C000615
PGDB_AS001212
View
% Degradation
-
=
75
%
10 nM
24 h
-
-
HL-60
CN117982498A
PGDB_A014956
PGDB_C000559
PGDB_AS001212
View
% Degradation
-
=
100
%
10 nM
24 h
-
-
HL-60
CN117982498A
PGDB_A016660
PGDB_C000608
PGDB_AS001212
View
% Degradation
-
=
47
%
10 nM
24 h
-
-
HL-60
CN117982498A
PGDB_A017628
PGDB_C000561
PGDB_AS001212
View
% Degradation
-
=
100
%
10 nM
24 h
-
-
HL-60
CN117982498A
PGDB_A018596
PGDB_C000636
PGDB_AS001212
View
% Degradation
-
=
100
%
10 nM
24 h
-
-
HL-60
CN117982498A
PGDB_A020836
PGDB_C000628
PGDB_AS001212
View
% Degradation
-
=
97
%
10 nM
24 h
-
-
HL-60
CN117982498A
PGDB_A021691
PGDB_C000541
PGDB_AS001212
View
% Degradation
-
=
100
%
10 nM
24 h
-
-
HL-60
CN117982498A
PGDB_A021807
PGDB_C000621
PGDB_AS001212
View
% Degradation
-
=
100
%
10 nM
24 h
-
-
HL-60
CN117982498A
PGDB_A023829
PGDB_C000607
PGDB_AS001212
View
% Degradation
-
=
93
%
10 nM
24 h
-
-
HL-60
CN117982498A
PGDB_A027887
PGDB_C000639
PGDB_AS001212
View
% Degradation
-
=
100
%
10 nM
24 h
-
-
HL-60
CN117982498A
PGDB_A029368
PGDB_C000606
PGDB_AS001212
View
% Degradation
-
=
99
%
10 nM
24 h
-
-
HL-60
CN117982498A
PGDB_A030794
PGDB_C000641
PGDB_AS001212
View
% Degradation
-
=
77
%
10 nM
24 h
-
-
HL-60
CN117982498A
PGDB_A034120
PGDB_C000562
PGDB_AS001212
View
% Degradation
-
=
100
%
10 nM
24 h
-
-
HL-60
CN117982498A
PGDB_A035399
PGDB_C000610
PGDB_AS001212
View
% Degradation
-
=
96
%
10 nM
24 h
-
-
HL-60
CN117982498A
PGDB_A035908
PGDB_C000554
PGDB_AS001212
View
% Degradation
-
=
98
%
10 nM
24 h
-
-
HL-60
CN117982498A
PGDB_A040540
PGDB_C000612
PGDB_AS001212
View
% Degradation
-
=
100
%
10 nM
24 h
-
-
HL-60
CN117982498A
PGDB_A040772
PGDB_C000629
PGDB_AS001212
View
% Degradation
-
=
71
%
10 nM
24 h
-
-
HL-60
CN117982498A
PGDB_A042299
PGDB_C000642
PGDB_AS001212
View
% Degradation
-
=
84
%
10 nM
24 h
-
-
HL-60
CN117982498A
PGDB_A043385
PGDB_C000540
PGDB_AS001212
View