PatGlueDB
Search
Browse
Statistics
Contact
Help
·
SIMM · NJU
Assay
PGDB_AS001227
System: cell_based
Target: KRAS
Assay context summary
Assay context
58 activity records
Assay family
% Degradation
System
cell_based
Readout
Dmax
Target
KRAS
E3
Not specified
Organism
Homo sapiens
Technology
luminescence
Activity compounds and values
Activity records
58 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Dmax
-
=
71
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A000080
PGDB_C031947
PGDB_AS001227
View
Dmax
-
=
82
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A000166
PGDB_C031975
PGDB_AS001227
View
Dmax
-
=
70
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A000488
PGDB_C031986
PGDB_AS001227
View
Dmax
-
=
89
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A000935
PGDB_C031973
PGDB_AS001227
View
Dmax
-
=
78
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A001137
PGDB_C031978
PGDB_AS001227
View
Dmax
-
=
82
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A001297
PGDB_C031991
PGDB_AS001227
View
Dmax
-
=
87
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A001460
PGDB_C031997
PGDB_AS001227
View
Dmax
-
=
58
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A001603
PGDB_C031948
PGDB_AS001227
View
Dmax
-
=
84
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A001635
PGDB_C031967
PGDB_AS001227
View
Dmax
-
=
81
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A001723
PGDB_C031981
PGDB_AS001227
View
Dmax
-
=
78
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A002020
PGDB_C031962
PGDB_AS001227
View
Dmax
-
=
85
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A002361
PGDB_C031951
PGDB_AS001227
View
Dmax
-
=
92
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A002509
PGDB_C031944
PGDB_AS001227
View
Dmax
-
=
90
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A002656
PGDB_C031996
PGDB_AS001227
View
Dmax
-
=
86
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A002772
PGDB_C031953
PGDB_AS001227
View
Dmax
-
=
82
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A002916
PGDB_C031958
PGDB_AS001227
View
Dmax
-
=
73
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A003149
PGDB_C031980
PGDB_AS001227
View
Dmax
-
=
85
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A003420
PGDB_C031977
PGDB_AS001227
View
Dmax
-
=
75
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A003544
PGDB_C031945
PGDB_AS001227
View
Dmax
-
=
85
%
-
18 h
KRAS
-
-
WO2026114958A1
PGDB_A003652
PGDB_C031994
PGDB_AS001227
View