Assay
PGDB_AS001243
System: cell_basedCell line: MM.1S
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 30 | nM | - | — | - | - | MM.1S | WO2023025136A1 | PGDB_A011009 | PGDB_C009601 | PGDB_AS001243 | View | |
| IC50 | - | = | 0.03 | nM | - | — | - | - | MM.1S | WO2023025136A1 | PGDB_A014969 | PGDB_C009997 | PGDB_AS001243 | View | |
| IC50 | - | = | 0.026 | nM | - | — | - | - | MM.1S | WO2023025136A1 | PGDB_A039973 | PGDB_C009985 | PGDB_AS001243 | View | |
| IC50 | - | = | 0.064 | nM | - | — | - | - | MM.1S | WO2023025136A1 | PGDB_A040190 | PGDB_C009999 | PGDB_AS001243 | View | |
| IC50 | - | = | 0.046 | nM | - | — | - | - | MM.1S | WO2023025136A1 | PGDB_A054605 | PGDB_C009989 | PGDB_AS001243 | View |