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SIMM · NJU
Assay
PGDB_AS001257
System: cell_based
Cell line: HEK293
Assay context summary
Assay context
82 activity records
Assay family
% Degradation
System
cell_based
Readout
Dmax
E3
Not specified
Cell line
HEK293
Organism
Homo sapiens
Technology
luminescence
Activity compounds and values
Activity records
82 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Dmax
-
=
-0.1
%
-
24 h
GSPT1
-
HEK293
WO2025224249A1
PGDB_A007405
PGDB_C011702
PGDB_AS001257
View
Dmax
-
=
10.1
%
-
24 h
GSPT1
-
HEK293
WO2025224249A1
PGDB_A008766
PGDB_C011719
PGDB_AS001257
View
Dmax
-
=
6.2
%
-
24 h
GSPT1
-
HEK293
WO2025224249A1
PGDB_A009045
PGDB_C011729
PGDB_AS001257
View
Dmax
-
=
31.5
%
-
24 h
GSPT1
-
HEK293
WO2025224249A1
PGDB_A009353
PGDB_C011750
PGDB_AS001257
View
Dmax
-
=
10.5
%
-
24 h
GSPT1
-
HEK293
WO2025224249A1
PGDB_A011478
PGDB_C011766
PGDB_AS001257
View
Dmax
-
=
11.2
%
-
24 h
GSPT1
-
HEK293
WO2025224249A1
PGDB_A011636
PGDB_C011751
PGDB_AS001257
View
Dmax
-
=
1.2
%
-
24 h
GSPT1
-
HEK293
WO2025224249A1
PGDB_A013425
PGDB_C011696
PGDB_AS001257
View
Dmax
-
=
9.1
%
-
24 h
GSPT1
-
HEK293
WO2025224249A1
PGDB_A015026
PGDB_C011703
PGDB_AS001257
View
Dmax
-
=
3.1
%
-
24 h
GSPT1
-
HEK293
WO2025224249A1
PGDB_A015233
PGDB_C011739
PGDB_AS001257
View
Dmax
-
=
4.8
%
-
24 h
GSPT1
-
HEK293
WO2025224249A1
PGDB_A015268
PGDB_C011772
PGDB_AS001257
View
Dmax
-
=
6.2
%
-
24 h
GSPT1
-
HEK293
WO2025224249A1
PGDB_A015601
PGDB_C011757
PGDB_AS001257
View
Dmax
-
=
5.1
%
-
24 h
GSPT1
-
HEK293
WO2025224249A1
PGDB_A017778
PGDB_C011762
PGDB_AS001257
View
Dmax
-
=
6.5
%
-
24 h
GSPT1
-
HEK293
WO2025224249A1
PGDB_A017976
PGDB_C011714
PGDB_AS001257
View
Dmax
-
=
4
%
-
24 h
GSPT1
-
HEK293
WO2025224249A1
PGDB_A018364
PGDB_C011700
PGDB_AS001257
View
Dmax
-
=
1.5
%
-
24 h
GSPT1
-
HEK293
WO2025224249A1
PGDB_A018779
PGDB_C011705
PGDB_AS001257
View
Dmax
-
=
9.8
%
-
24 h
GSPT1
-
HEK293
WO2025224249A1
PGDB_A019137
PGDB_C011721
PGDB_AS001257
View
Dmax
-
=
2.6
%
-
24 h
GSPT1
-
HEK293
WO2025224249A1
PGDB_A019138
PGDB_C011732
PGDB_AS001257
View
Dmax
-
=
5.1
%
-
24 h
GSPT1
-
HEK293
WO2025224249A1
PGDB_A019941
PGDB_C011716
PGDB_AS001257
View
Dmax
-
=
5.3
%
-
24 h
GSPT1
-
HEK293
WO2025224249A1
PGDB_A020529
PGDB_C011717
PGDB_AS001257
View
Dmax
-
=
3.7
%
-
24 h
GSPT1
-
HEK293
WO2025224249A1
PGDB_A021485
PGDB_C011734
PGDB_AS001257
View