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Compound
PGDB_C011757
3 activity records1 related patents
2D structure
Cc1cc(C2CCC(=O)NC2=O)ccc1N1C[C@H](Nc2nnc(C34CC(C(F)(F)F)(C3)C4)o2)[C@H]1CCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 6.2 | % | - | 24 h | GSPT1 | - | HEK293 | WO2025224249A1 | PGDB_A015601 | PGDB_C011757 | PGDB_AS001257 | View |
| DC50 | - | = | 140.4 | nM | - | — | CDK2 | - | HEK293 | WO2025224249A1 | PGDB_A036223 | PGDB_C011757 | PGDB_AS000391 | View |
| Dmax | - | = | 62.2 | % | - | 24 h | CDK2 | - | HEK293 | WO2025224249A1 | PGDB_A073034 | PGDB_C011757 | PGDB_AS002358 | View |