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SIMM · NJU
Assay
PGDB_AS001306
System: cell_based
Target: GSPT1
Cell line: GP2D
Assay context summary
Assay context
12 activity records
Assay family
viability
System
cell_based
Readout
Fold change
Target
GSPT1
E3
Not specified
Cell line
GP2D
Organism
Homo sapiens
Technology
CCK-8
Detection target
cell_proliferation
Activity compounds and values
Activity records
12 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Potency ratio
Ref1
=
2-10
fold
-
—
GSPT1
-
GP2D
WO2025026218A1
PGDB_A009539
PGDB_C005374
PGDB_AS001306
View
Potency ratio
Ref1
=
0-1.3
fold
-
—
GSPT1
-
GP2D
WO2025026218A1
PGDB_A019882
PGDB_C005378
PGDB_AS001306
View
Potency ratio
Ref1
=
10-20
fold
-
—
GSPT1
-
GP2D
WO2025026218A1
PGDB_A026196
PGDB_C005376
PGDB_AS001306
View
Potency ratio
Ref1
=
2-10
fold
-
—
GSPT1
-
GP2D
WO2025026218A1
PGDB_A029334
PGDB_C005373
PGDB_AS001306
View
Potency ratio
Ref1
=
2-10
fold
-
—
GSPT1
-
GP2D
WO2025026218A1
PGDB_A046023
PGDB_C005383
PGDB_AS001306
View
Potency ratio
Ref1
=
1.3-2
fold
-
—
GSPT1
-
GP2D
WO2025026218A1
PGDB_A054222
PGDB_C005379
PGDB_AS001306
View
Potency ratio
Ref1
=
20-30
fold
-
—
GSPT1
-
GP2D
WO2025026218A1
PGDB_A058371
PGDB_C005375
PGDB_AS001306
View
Potency ratio
Ref1
=
2-10
fold
-
—
GSPT1
-
GP2D
WO2025026218A1
PGDB_A062994
PGDB_C005380
PGDB_AS001306
View
Potency ratio
Ref1
=
2-10
fold
-
—
GSPT1
-
GP2D
WO2025026218A1
PGDB_A063503
PGDB_C005382
PGDB_AS001306
View
Potency ratio
Ref1
=
2-10
fold
-
—
GSPT1
-
GP2D
WO2025026218A1
PGDB_A064069
PGDB_C005384
PGDB_AS001306
View
Potency ratio
Ref1
>=
30
fold
-
—
GSPT1
-
GP2D
WO2025026218A1
PGDB_A072724
PGDB_C005381
PGDB_AS001306
View
Potency ratio
Ref1
=
2-10
fold
-
—
GSPT1
-
GP2D
WO2025026218A1
PGDB_A076386
PGDB_C005377
PGDB_AS001306
View