Assay
PGDB_AS001375
System: cell_basedCell line: MV-4-11
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 1 | nM | - | — | GSPT1 | - | MV-4-11 | WO2024222918A1 | PGDB_A021085 | PGDB_C003265 | PGDB_AS001375 | View | |
| IC50 | - | >= | 1000 | nM | - | — | GSPT1 | - | MV-4-11 | WO2024222918A1 | PGDB_A021484 | PGDB_C003267 | PGDB_AS001375 | View | |
| IC50 | - | = | 1-10 | nM | - | — | GSPT1 | - | MV-4-11 | WO2024222918A1 | PGDB_A021626 | PGDB_C003262 | PGDB_AS001375 | View | |
| IC50 | - | = | 10-100 | nM | - | — | GSPT1 | - | MV-4-11 | WO2024222918A1 | PGDB_A041170 | PGDB_C003219 | PGDB_AS001375 | View | |
| IC50 | - | = | 10-100 | nM | - | — | GSPT1 | - | MV-4-11 | WO2024222918A1 | PGDB_A042018 | PGDB_C003266 | PGDB_AS001375 | View | |
| IC50 | - | = | 10-100 | nM | - | — | GSPT1 | - | MV-4-11 | WO2024222918A1 | PGDB_A045867 | PGDB_C000059 | PGDB_AS001375 | View | |
| IC50 | - | = | 10-100 | nM | - | — | GSPT1 | - | MV-4-11 | WO2024222918A1 | PGDB_A049914 | PGDB_C003237 | PGDB_AS001375 | View | |
| IC50 | - | = | 10-100 | nM | - | — | GSPT1 | - | MV-4-11 | WO2024222918A1 | PGDB_A070467 | PGDB_C003221 | PGDB_AS001375 | View |