Assay
PGDB_AS001400
System: cell_basedCell line: MDA-MB-231
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 50-100 | nM | - | — | ESR1 | - | MDA-MB-231 | CN116239566A | PGDB_A008855 | PGDB_C025816 | PGDB_AS001400 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | MDA-MB-231 | CN116239566A | PGDB_A024516 | PGDB_C025824 | PGDB_AS001400 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | MDA-MB-231 | CN116239566A | PGDB_A037894 | PGDB_C019597 | PGDB_AS001400 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | MDA-MB-231 | CN116239566A | PGDB_A039063 | PGDB_C025818 | PGDB_AS001400 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | MDA-MB-231 | CN116239566A | PGDB_A039507 | PGDB_C025823 | PGDB_AS001400 | View | |
| IC50 | - | = | 50-100 | nM | - | — | ESR1 | - | MDA-MB-231 | CN116239566A | PGDB_A046651 | PGDB_C025822 | PGDB_AS001400 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | MDA-MB-231 | CN116239566A | PGDB_A062211 | PGDB_C025826 | PGDB_AS001400 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | MDA-MB-231 | CN116239566A | PGDB_A071684 | PGDB_C019596 | PGDB_AS001400 | View |