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Compound
PGDB_C025822
10 activity records1 related patents
2D structure
O=C1CCC(N2Cc3cc(CN4CCN(c5ccc(C(=C(CCCl)c6ccccc6)c6ccccc6)cc5)CC4)ccc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 50-100 | nM | - | — | ESR1 | - | MM.1S | CN116239566A | PGDB_A027517 | PGDB_C025822 | PGDB_AS001148 | View |
| IC50 | - | = | 100-500 | nM | - | — | ESR1 | - | Hep3B2.7-1 | CN116239566A | PGDB_A029153 | PGDB_C025822 | PGDB_AS000032 | View |
| IC50 | - | = | 100-500 | nM | - | — | ESR1 | - | SU-DHL-6 | CN116239566A | PGDB_A030640 | PGDB_C025822 | PGDB_AS002532 | View |
| IC50 | - | = | 50-100 | nM | - | — | ESR1 | - | HCC827 | CN116239566A | PGDB_A032650 | PGDB_C025822 | PGDB_AS001534 | View |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | Kasumi-1 | CN116239566A | PGDB_A033604 | PGDB_C025822 | PGDB_AS000517 | View |
| IC50 | - | = | 50-100 | nM | - | — | ESR1 | - | T47D | CN116239566A | PGDB_A045060 | PGDB_C025822 | PGDB_AS000239 | View |
| IC50 | - | = | 50-100 | nM | - | — | ESR1 | - | SW620 | CN116239566A | PGDB_A045847 | PGDB_C025822 | PGDB_AS001305 | View |
| IC50 | - | = | 50-100 | nM | - | — | ESR1 | - | MDA-MB-231 | CN116239566A | PGDB_A046651 | PGDB_C025822 | PGDB_AS001400 | View |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | Mino | CN116239566A | PGDB_A065402 | PGDB_C025822 | PGDB_AS001392 | View |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | CCRF-CEM | CN116239566A | PGDB_A075728 | PGDB_C025822 | PGDB_AS000150 | View |