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O=C1CCC(N2Cc3cc(CN4CCN(c5ccc(C(=C(CCCl)c6ccc(O)cc6)c6ccc(O)cc6)cc5)CC4)ccc3C2=O)C(=O)N1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | SW620 | CN116239566A | PGDB_A017356 | PGDB_C025818 | PGDB_AS001305 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | CCRF-CEM | CN116239566A | PGDB_A018027 | PGDB_C025818 | PGDB_AS000150 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | T47D | CN116239566A | PGDB_A037030 | PGDB_C025818 | PGDB_AS000239 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | MDA-MB-231 | CN116239566A | PGDB_A039063 | PGDB_C025818 | PGDB_AS001400 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | HCC827 | CN116239566A | PGDB_A050070 | PGDB_C025818 | PGDB_AS001534 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | Mino | CN116239566A | PGDB_A051850 | PGDB_C025818 | PGDB_AS001392 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | SU-DHL-6 | CN116239566A | PGDB_A056628 | PGDB_C025818 | PGDB_AS002532 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | MM.1S | CN116239566A | PGDB_A068824 | PGDB_C025818 | PGDB_AS001148 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | Hep3B2.7-1 | CN116239566A | PGDB_A074282 | PGDB_C025818 | PGDB_AS000032 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | Kasumi-1 | CN116239566A | PGDB_A074337 | PGDB_C025818 | PGDB_AS000517 | View |