Assay

PGDB_AS001405

System: cell_basedTarget: CRBN
Assay context summary

Assay context

406 activity records
Assay familybiochemical
Systemcell_based
Readout% Inhibition
TargetCRBN
E3CRBN
OrganismHomo sapiens
TechnologyHTRF
Detection targetcell_inhibition
Activity compounds and values

Activity records

406 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C022400
% Inhibition-=53-60%0.5 uM3 hCRBNCRBN-CN119654316APGDB_A081918PGDB_C022400PGDB_AS001405View
2D structure for PGDB_C022039
% Inhibition-=40-53%0.5 uM3 hCRBNCRBN-CN119654316APGDB_A081924PGDB_C022039PGDB_AS001405View
2D structure for PGDB_C022360
% Inhibition-=53-60%0.5 uM3 hCRBNCRBN-CN119654316APGDB_A081929PGDB_C022360PGDB_AS001405View
2D structure for PGDB_C022170
% Inhibition-=53-60%0.5 uM3 hCRBNCRBN-CN119654316APGDB_A081931PGDB_C022170PGDB_AS001405View
2D structure for PGDB_C021998
% Inhibition-=30-40%0.5 uM3 hCRBNCRBN-CN119654316APGDB_A081934PGDB_C021998PGDB_AS001405View
2D structure for PGDB_C022093
% Inhibition-=53-60%0.5 uM3 hCRBNCRBN-CN119654316APGDB_A081937PGDB_C022093PGDB_AS001405View
2D structure for PGDB_C022059
% Inhibition-=20-30%0.5 uM3 hCRBNCRBN-CN119654316APGDB_A081962PGDB_C022059PGDB_AS001405View
2D structure for PGDB_C022091
% Inhibition-=53-60%0.5 uM3 hCRBNCRBN-CN119654316APGDB_A081968PGDB_C022091PGDB_AS001405View
2D structure for PGDB_C022232
% Inhibition-=53-60%0.5 uM3 hCRBNCRBN-CN119654316APGDB_A081972PGDB_C022232PGDB_AS001405View
2D structure for PGDB_C022331
% Inhibition-=30-40%0.5 uM3 hCRBNCRBN-CN119654316APGDB_A081976PGDB_C022331PGDB_AS001405View
2D structure for PGDB_C022282
% Inhibition-=40-53%0.5 uM3 hCRBNCRBN-CN119654316APGDB_A081995PGDB_C022282PGDB_AS001405View
2D structure for PGDB_C022261
% Inhibition-=53-60%0.5 uM3 hCRBNCRBN-CN119654316APGDB_A082001PGDB_C022261PGDB_AS001405View
2D structure for PGDB_C022104
% Inhibition-=53-60%0.5 uM3 hCRBNCRBN-CN119654316APGDB_A082025PGDB_C022104PGDB_AS001405View
2D structure for PGDB_C022105
% Inhibition-=40-53%0.5 uM3 hCRBNCRBN-CN119654316APGDB_A082058PGDB_C022105PGDB_AS001405View
2D structure for PGDB_C022157
% Inhibition-=53-60%0.5 uM3 hCRBNCRBN-CN119654316APGDB_A082064PGDB_C022157PGDB_AS001405View
2D structure for PGDB_C022382
% Inhibition-=20-30%0.5 uM3 hCRBNCRBN-CN119654316APGDB_A082066PGDB_C022382PGDB_AS001405View
2D structure for PGDB_C022148
% Inhibition-=30-40%0.5 uM3 hCRBNCRBN-CN119654316APGDB_A082069PGDB_C022148PGDB_AS001405View
2D structure for PGDB_C022097
% Inhibition-=30-40%0.5 uM3 hCRBNCRBN-CN119654316APGDB_A082071PGDB_C022097PGDB_AS001405View
2D structure for PGDB_C022399
% Inhibition-=53-60%0.5 uM3 hCRBNCRBN-CN119654316APGDB_A082076PGDB_C022399PGDB_AS001405View
2D structure for PGDB_C022146
% Inhibition-=20-30%0.5 uM3 hCRBNCRBN-CN119654316APGDB_A082082PGDB_C022146PGDB_AS001405View
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