PatGlueDB
Search
Browse
Statistics
Contact
Help
·
SIMM · NJU
Assay
PGDB_AS001415
System: cell_based
Target: CDK2
Cell line: HEK293
Assay context summary
Assay context
45 activity records
Assay family
% Degradation
System
cell_based
Readout
Dmax
Target
CDK2
E3
Not specified
Cell line
HEK293
Organism
Homo sapiens
Technology
luminescence
Activity compounds and values
Activity records
45 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Dmax
-
>
80
%
30 uM
24 h
CDK2
-
HEK293
WO2025224262A1
PGDB_A011720
PGDB_C027528
PGDB_AS001415
View
Dmax
-
>
80
%
30 uM
24 h
CDK2
-
HEK293
WO2025224262A1
PGDB_A012797
PGDB_C027542
PGDB_AS001415
View
Dmax
-
>
80
%
30 uM
24 h
CDK2
-
HEK293
WO2025224262A1
PGDB_A013708
PGDB_C027508
PGDB_AS001415
View
Dmax
-
>
80
%
30 uM
24 h
CDK2
-
HEK293
WO2025224262A1
PGDB_A013788
PGDB_C027498
PGDB_AS001415
View
Dmax
-
>
80
%
30 uM
24 h
CDK2
-
HEK293
WO2025224262A1
PGDB_A014212
PGDB_C011831
PGDB_AS001415
View
Dmax
-
>
80
%
30 uM
24 h
CDK2
-
HEK293
WO2025224262A1
PGDB_A014713
PGDB_C027501
PGDB_AS001415
View
Dmax
-
>
80
%
30 uM
24 h
CDK2
-
HEK293
WO2025224262A1
PGDB_A016442
PGDB_C011773
PGDB_AS001415
View
Dmax
-
>
80
%
30 uM
24 h
CDK2
-
HEK293
WO2025224262A1
PGDB_A019875
PGDB_C027478
PGDB_AS001415
View
Dmax
-
>
80
%
30 uM
24 h
CDK2
-
HEK293
WO2025224262A1
PGDB_A024693
PGDB_C027540
PGDB_AS001415
View
Dmax
-
>
80
%
30 uM
24 h
CDK2
-
HEK293
WO2025224262A1
PGDB_A025560
PGDB_C027547
PGDB_AS001415
View
Dmax
-
>
80
%
30 uM
24 h
CDK2
-
HEK293
WO2025224262A1
PGDB_A030144
PGDB_C027461
PGDB_AS001415
View
Dmax
-
>
80
%
30 uM
24 h
CDK2
-
HEK293
WO2025224262A1
PGDB_A034780
PGDB_C027505
PGDB_AS001415
View
Dmax
-
>
80
%
30 uM
24 h
CDK2
-
HEK293
WO2025224262A1
PGDB_A036574
PGDB_C027538
PGDB_AS001415
View
Dmax
-
>
80
%
30 uM
24 h
CDK2
-
HEK293
WO2025224262A1
PGDB_A036717
PGDB_C027459
PGDB_AS001415
View
Dmax
-
>
80
%
30 uM
24 h
CDK2
-
HEK293
WO2025224262A1
PGDB_A037013
PGDB_C027460
PGDB_AS001415
View
Dmax
-
>
80
%
30 uM
24 h
CDK2
-
HEK293
WO2025224262A1
PGDB_A037592
PGDB_C027546
PGDB_AS001415
View
Dmax
-
>
80
%
30 uM
24 h
CDK2
-
HEK293
WO2025224262A1
PGDB_A037650
PGDB_C011847
PGDB_AS001415
View
Dmax
-
>
80
%
30 uM
24 h
CDK2
-
HEK293
WO2025224262A1
PGDB_A039680
PGDB_C027499
PGDB_AS001415
View
Dmax
-
>
80
%
30 uM
24 h
CDK2
-
HEK293
WO2025224262A1
PGDB_A040815
PGDB_C027541
PGDB_AS001415
View
Dmax
-
>
80
%
30 uM
24 h
CDK2
-
HEK293
WO2025224262A1
PGDB_A041019
PGDB_C027497
PGDB_AS001415
View